# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | DS-1971a | rac-6o | t1/2 | = | 2.8 | min | ALA4623859 | hr | Mus musculus | |||
2. | DS-1971a | rac-6o | IC50 | = | 59.4 | nM | ALA4623855 | 7.23 | nM | Mus musculus | ||
3. | DS-1971a | rac-6o | INH | = | 81.9 | % | ALA4623841 | % | Mus musculus | |||
4. | ALA4639987 | rac-6q | IC50 | = | 15 | nM | ALA4623821 | 7.82 | nM | Mus musculus | ||
5. | ALA4637488 | rac-6p | IC50 | = | 28 | nM | ALA4623821 | 7.55 | nM | Mus musculus | ||
6. | DS-1971a | rac-6o | IC50 | = | 56.3 | nM | ALA4623821 | 7.25 | nM | Mus musculus | ||
7. | DS-1971a | rac-6o | IC50 | = | 26.5 | nM | ALA4623821 | 7.58 | nM | Mus musculus | ||
8. | ALA4637909 | rac-6n | IC50 | = | 28 | nM | ALA4623821 | 7.55 | nM | Mus musculus | ||
9. | ALA4642940 | rac-6m | IC50 | = | 41 | nM | ALA4623821 | 7.39 | nM | Mus musculus | ||
10. | ALA4648397 | rac-6l | IC50 | = | 56 | nM | ALA4623821 | 7.25 | nM | Mus musculus | ||
11. | ALA4645788 | rac-6k | IC50 | = | 96 | nM | ALA4623821 | 7.02 | nM | Mus musculus | ||
12. | ALA4648771 | rac-6j | IC50 | = | 2800 | nM | ALA4623821 | 5.55 | nM | Mus musculus | ||
13. | ALA4647897 | rac-6i | IC50 | 0 | ALA4623821 | Not Determined | Mus musculus | |||||
14. | ALA4640756 | rac-6h | IC50 | = | 400 | nM | ALA4623821 | 6.40 | nM | Mus musculus | ||
15. | ALA4642726 | rac-6g | IC50 | = | 1300 | nM | ALA4623821 | 5.89 | nM | Mus musculus | ||
16. | ALA4635030 | rac-6f | IC50 | = | 2800 | nM | ALA4623821 | 5.55 | nM | Mus musculus | ||
17. | ALA4633573 | rac-6e | IC50 | = | 100 | nM | ALA4623821 | 7.00 | nM | Mus musculus | ||
18. | ALA4641238 | rac-6d | IC50 | 0 | ALA4623821 | Not Determined | Mus musculus | |||||
19. | ALA4642571 | rac-6c | IC50 | = | 17 | nM | ALA4623821 | 7.77 | nM | Mus musculus | ||
20. | ALA4632675 | rac-6b | IC50 | = | 240 | nM | ALA4623821 | 6.62 | nM | Mus musculus |