# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4210512 | (R/S)-ND-336 | INH | = | 31 | % | ALA4201805 | % | Homo sapiens | |||
2. | ALA4214929 | (S)-ND-336 | INH | = | 25 | % | ALA4201805 | % | Homo sapiens | |||
3. | ALA4215451 | (R)-2; (R)-ND-336 | INH | = | 41 | % | ALA4201805 | % | Homo sapiens | |||
4. | ALA4208519 | 26f | IC50 | = | 0.48 | uM | ALA4186131 | 6.32 | nM | Homo sapiens | ||
5. | ALA4215407 | 26a | IC50 | = | 0.09 | uM | ALA4186131 | 7.05 | nM | Homo sapiens | ||
6. | ALA4167357 | 2 | INH | = | 15 | % | ALA4151334 | % | Homo sapiens | |||
7. | ALA497985 | 51 | Ki | = | 2200 | nM | ALA4151326 | 5.66 | nM | Homo sapiens | ||
8. | ALA4873384 | (R)-18 | IC50 | = | 8.448 | uM | ALA4835179 | 5.07 | nM | Homo sapiens | ||
9. | ALA4854306 | 29 | IC50 | > | 3 | uM | ALA4835179 | nM | Homo sapiens | |||
10. | ALA4102106 | 31g | IC50 | > | 10 | uM | ALA4010775 | nM | Homo sapiens | |||
11. | apratastat | 5h | IC50 | = | 85 | nM | ALA3888620 | 7.07 | 411136 | nM | Homo sapiens | |
12. | ALA3648907 | BDBM113593 | IC50 | > | 10000 | nM | ALA3888620 | 411135 | nM | Homo sapiens | ||
13. | ALA3648906 | BDBM113592 | IC50 | > | 10000 | nM | ALA3888620 | 411134 | nM | Homo sapiens | ||
14. | ALA3648905 | BDBM113591 | IC50 | > | 10000 | nM | ALA3888620 | 411133 | nM | Homo sapiens | ||
15. | ALA3648904 | BDBM113590 | IC50 | > | 10000 | nM | ALA3888620 | 411132 | nM | Homo sapiens | ||
16. | ALA3959985 | BDBM235932 | IC50 | > | 10000 | nM | ALA3888620 | 411131 | nM | Homo sapiens | ||
17. | ALA3648903 | BDBM113589 | IC50 | = | 3054 | nM | ALA3888620 | 5.51 | 411130 | nM | Homo sapiens | |
18. | ALA3648902 | BDBM113588 | IC50 | = | 9254 | nM | ALA3888620 | 5.03 | 411129 | nM | Homo sapiens | |
19. | ALA3648893 | BDBM113577 | IC50 | > | 10000 | nM | ALA3888620 | 411128 | nM | Homo sapiens | ||
20. | apratastat | 5h | IC50 | = | 85 | nM | ALA3888014 | 7.07 | 367348 | nM | Homo sapiens |