# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | JNJ-42226314 | BDBM150300 | Inhibition | = | 4 | % | ALA5305002 | % | Homo sapiens | |||
2. | ALA3585742 | 17a | IC50 | = | 100 | uM | ALA3803181 | 4.00 | nM | Homo sapiens | ||
3. | ALA3799135 | 19a | IC50 | = | 25 | uM | ALA3803181 | 4.60 | nM | Homo sapiens | ||
4. | ALA3799329 | 19b | IC50 | = | 45 | uM | ALA3803181 | 4.35 | nM | Homo sapiens | ||
5. | ALA3800112 | 19c | IC50 | = | 19 | uM | ALA3803181 | 4.72 | nM | Homo sapiens | ||
6. | ALA3799182 | 19d | IC50 | = | 12 | uM | ALA3803181 | 4.92 | nM | Homo sapiens | ||
7. | ALA3799525 | 19e | IC50 | = | 11 | uM | ALA3803181 | 4.96 | nM | Homo sapiens | ||
8. | ALA3800020 | 19f | IC50 | = | 19 | uM | ALA3803181 | 4.72 | nM | Homo sapiens | ||
9. | ALA3797774 | 19g | IC50 | = | 28 | uM | ALA3803181 | 4.55 | nM | Homo sapiens | ||
10. | ALA3799985 | 19h | IC50 | = | 4.9 | uM | ALA3803181 | 5.31 | nM | Homo sapiens | ||
11. | ALA3798282 | 19i | IC50 | = | 6.7 | uM | ALA3803181 | 5.17 | nM | Homo sapiens | ||
12. | ALA3800401 | 19j | IC50 | = | 7.7 | uM | ALA3803181 | 5.11 | nM | Homo sapiens | ||
13. | ALA3781319 | (S)-24 | Ki | = | 12540 | nM | ALA3783218 | 4.90 | nM | Homo sapiens | ||
14. | ALA3781788 | (S)-17 | Ki | > | 22100 | nM | ALA3783218 | nM | Homo sapiens | |||
15. | ALA3780324 | (S)-10 | Ki | > | 22100 | nM | ALA3783218 | nM | Homo sapiens | |||
16. | ALA3393386 | (S)-23 | Ki | > | 22100 | nM | ALA3783218 | nM | Homo sapiens | |||
17. | ALA3770794 | 2b | IC50 | > | 10 | uM | ALA3772683 | nM | Homo sapiens | |||
18. | ALA3771081 | 2a | IC50 | > | 10 | uM | ALA3772683 | nM | Homo sapiens | |||
19. | ALA3769636 | 1i | IC50 | > | 10 | uM | ALA3772683 | nM | Homo sapiens | |||
20. | ALA238913 | 7c | IC50 | = | 6.2 | uM | ALA3772683 | 5.21 | nM | Homo sapiens |