# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Retigabine | 1 (Retigabine) | Activity | = | 3.04 | ALA5151183 | Homo sapiens | |||||
2. | Retigabine | 1 (Retigabine) | Activity | = | 0.09 | mV | ALA5151182 | mV | Homo sapiens | |||
3. | ALA5180351 | L3-14; HN37 | Activity | = | 3.14 | ALA5151181 | Homo sapiens | |||||
4. | ALA5180351 | L3-14; HN37 | Activity | = | -9.03 | mV | ALA5151180 | mV | Homo sapiens | |||
5. | ALA5178988 | CLE030 | EC50 | = | 4.5 | uM | ALA5125932 | 5.35 | nM | Homo sapiens | ||
6. | ALA4549229 | RL-24 | EC50 | = | 0.54 | uM | ALA5116584 | 6.27 | nM | Homo sapiens | ||
7. | ALA5185685 | RL-71 | EC50 | = | 1.06 | uM | ALA5116584 | 5.97 | nM | Homo sapiens | ||
8. | ALA4458793 | RL-56 | EC50 | = | 3.78 | uM | ALA5116584 | 5.42 | nM | Homo sapiens | ||
9. | ALA5200636 | RL-15 | EC50 | = | 3.78 | uM | ALA5116584 | 5.42 | nM | Homo sapiens | ||
10. | Retigabine | 1 (Retigabine) | EC50 | = | 0.8 | uM | ALA4403832 | 6.10 | nM | Homo sapiens | ||
11. | ALA4457044 | 24a | EC50 | = | 0.35 | uM | ALA4403832 | 6.46 | nM | Homo sapiens | ||
12. | ALA4545892 | 23a | EC50 | = | 1.07 | uM | ALA4403832 | 5.97 | nM | Homo sapiens | ||
13. | Retigabine | 1 (Retigabine) | Activity | = | -21.95 | mV | ALA4403828 | mV | Homo sapiens | |||
14. | ALA4457044 | 24a | Activity | = | -19.7 | mV | ALA4403828 | mV | Homo sapiens | |||
15. | ALA4545892 | 23a | Activity | = | -25.6 | mV | ALA4403828 | mV | Homo sapiens | |||
16. | Retigabine | 1 (Retigabine) | EC50 | = | 3.45 | uM | ALA4385397 | 5.46 | nM | Homo sapiens | ||
17. | ALA4438770 | 13 | EC50 | = | 1.37 | uM | ALA4385397 | 5.86 | nM | Homo sapiens | ||
18. | retigabine derivative 10g | 10g | EC50 | = | 1.68 | uM | ALA4385397 | 5.78 | nM | Homo sapiens | ||
19. | ALA4450214 | 8g | EC50 | = | 2.43 | uM | ALA4385397 | 5.61 | nM | Homo sapiens | ||
20. | ALA4448132 | 6e | Ratio | = | 4.8 | ALA4385395 | Homo sapiens |