# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MaxiPost | (S)-(+)-1 | EC50 | = | 2.4 | uM | ALA2327422 | 5.62 | nM | Homo sapiens | ||
2. | Retigabine | 1 (Retigabine) | EC50 | = | 0.8 | uM | ALA4403832 | 6.10 | nM | Homo sapiens | ||
3. | ALA4457044 | 24a | EC50 | = | 0.35 | uM | ALA4403832 | 6.46 | nM | Homo sapiens | ||
4. | ALA4545892 | 23a | EC50 | = | 1.07 | uM | ALA4403832 | 5.97 | nM | Homo sapiens | ||
5. | Retigabine | 1 (Retigabine) | Activity | = | -21.95 | mV | ALA4403828 | mV | Homo sapiens | |||
6. | ALA4457044 | 24a | Activity | = | -19.7 | mV | ALA4403828 | mV | Homo sapiens | |||
7. | ALA4545892 | 23a | Activity | = | -25.6 | mV | ALA4403828 | mV | Homo sapiens | |||
8. | Retigabine | 1 (Retigabine) | EC50 | = | 3.45 | uM | ALA4385397 | 5.46 | nM | Homo sapiens | ||
9. | ALA4438770 | 13 | EC50 | = | 1.37 | uM | ALA4385397 | 5.86 | nM | Homo sapiens | ||
10. | retigabine derivative 10g | 10g | EC50 | = | 1.68 | uM | ALA4385397 | 5.78 | nM | Homo sapiens | ||
11. | ALA4450214 | 8g | EC50 | = | 2.43 | uM | ALA4385397 | 5.61 | nM | Homo sapiens | ||
12. | ALA4448132 | 6e | Ratio | = | 4.8 | ALA4385395 | Homo sapiens | |||||
13. | ALA4438770 | 13 | Ratio | = | 4.59 | ALA4385384 | Homo sapiens | |||||
14. | ALA4562549 | 10h | Ratio | = | 2.57 | ALA4385384 | Homo sapiens | |||||
15. | retigabine derivative 10g | 10g | Ratio | = | 4.58 | ALA4385384 | Homo sapiens | |||||
16. | ALA4447666 | 10f | Ratio | = | 4.84 | ALA4385384 | Homo sapiens | |||||
17. | ALA4450990 | 10e | Ratio | = | 3.62 | ALA4385384 | Homo sapiens | |||||
18. | ALA4543293 | 10d | Ratio | = | 5.71 | ALA4385384 | Homo sapiens | |||||
19. | ALA4584514 | 10c | Ratio | = | 5.81 | ALA4385384 | Homo sapiens | |||||
20. | ALA4540288 | 10b | Ratio | = | 4.67 | ALA4385384 | Homo sapiens |