# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4752133 | 2 | Km | = | 86.55 | umol/L | ALA4672288 | nM | Homo sapiens | |||
2. | ALA4788098 | 1 | Km | = | 54.12 | umol/L | ALA4672288 | nM | Homo sapiens | |||
3. | ALA3780541 | SYL930 | Km | = | 42.62 | umol/L | ALA4672288 | nM | Homo sapiens | |||
4. | Fingolimod HCl | FTY720 (1a) | Km | = | 23.7 | umol/L | ALA4672288 | nM | Homo sapiens | |||
5. | ALA4752133 | 2 | Vmax | = | 2.15 | pmol/min | ALA4672287 | pmol/min | Homo sapiens | |||
6. | ALA4788098 | 1 | Vmax | = | 2.63 | pmol/min | ALA4672287 | pmol/min | Homo sapiens | |||
7. | ALA3780541 | SYL930 | Vmax | = | 0.53 | pmol/min | ALA4672287 | pmol/min | Homo sapiens | |||
8. | Fingolimod HCl | FTY720 (1a) | Vmax | = | 0.31 | pmol/min | ALA4672287 | pmol/min | Homo sapiens | |||
9. | ALA4752133 | 2 | CL | = | 0.025 | uL/min | ALA4672286 | uL/min | Homo sapiens | |||
10. | ALA4788098 | 1 | CL | = | 0.049 | uL/min | ALA4672286 | uL/min | Homo sapiens | |||
11. | ALA3780541 | SYL930 | CL | = | 0.012 | uL/min | ALA4672286 | uL/min | Homo sapiens | |||
12. | Fingolimod HCl | FTY720 (1a) | CL | = | 0.013 | uL/min | ALA4672286 | uL/min | Homo sapiens | |||
13. | ALA552462 | 5p | Activity | 0 | ALA4669302 | Active | Homo sapiens | |||||
14. | ALA1233528 | VOLASERTIB | Activity | 0 | ALA4669301 | Active | Homo sapiens | |||||
15. | ALA228814 | 1 | Activity | 0 | ALA4669300 | Active | Homo sapiens | |||||
16. | ABC294640 | ABC294640 | Activity | 0 | ALA4669299 | Active | Homo sapiens | |||||
17. | ABC294640 | ABC294640 | Activity | 0 | ALA4669298 | Active | Homo sapiens | |||||
18. | ABC294640 | ABC294640 | Activity | 0 | ALA4669297 | Active | Homo sapiens | |||||
19. | ALA552462 | 5p | Activity | = | 4.7 | pmol | ALA4669286 | pmol | Homo sapiens | |||
20. | ALA552462 | 5p | Activity | = | 87 | pmol | ALA4669285 | pmol | Homo sapiens |