# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AM-1638 | 21, AM-1638 | INH | = | 89 | % | ALA4388837 | % | Homo sapiens | |||
2. | ALA4460352 | 4 | EC50 | = | 240 | nM | ALA4351154 | 6.62 | nM | Homo sapiens | ||
3. | ALA4459769 | 3 | EC50 | = | 310 | nM | ALA4351154 | 6.51 | nM | Homo sapiens | ||
4. | ALA2096803 | 3 | EC50 | = | 290 | nM | ALA4351154 | 6.54 | nM | Homo sapiens | ||
5. | ALA4459895 | 22 | INH | 0 | ALA4341522 | Active | % | Homo sapiens | ||||
6. | ALA4748253 | 9 | INH | = | 89.2 | % | ALA4667700 | % | Homo sapiens | |||
7. | ALA4784899 | 51 | INH | = | 17.5 | % | ALA4667700 | % | Homo sapiens | |||
8. | ALA4789469 | 26 | INH | = | -13.5 | % | ALA4667700 | % | Homo sapiens | |||
9. | THPP-1 | THPP-1 | % inhibition | -5 | % | ALA4882952 | Not Active | % | Homo sapiens | |||
10. | MLi-2 | 1; MLi-2 | % inhibition | 5 | % | ALA4882952 | Not Active | % | Homo sapiens | |||
11. | ALA4866278 | 33 | INH | 0 | ALA4818053 | Not Active | % | Homo sapiens | ||||
12. | ALA4438921 | 132d | IC50 | = | 3 | uM | ALA4613582 | 5.52 | nM | Homo sapiens | ||
13. | ALA4634634 | 29 | INH | = | 2 | % | ALA4603428 | % | Homo sapiens | |||
14. | ALA1563898 | SID49679877 | AC50 | > | 70 | uM | ALA3214889 | inactive | nM | Homo sapiens | ||
15. | ALA1380801 | SID26725675 | AC50 | = | 17.43 | uM | ALA3214889 | 4.76 | active | nM | Homo sapiens | |
16. | ALA1475961 | SID57260543 | AC50 | = | 27.16 | uM | ALA3214889 | 4.57 | active | nM | Homo sapiens | |
17. | Isoquinoline-1,3(2H,4H)-dione | 5, ZINC-1601221 | AC50 | = | 1.34 | uM | ALA3214889 | 5.87 | active | nM | Homo sapiens | |
18. | N-[4-hydroxy-3-(1H-1,2,4-triazol-5-ylsulfanyl)naphthalen-1-yl]-4-methoxybenzenesulfonamide | SID16952410 | AC50 | = | 31.59 | uM | ALA3214889 | 4.50 | active | nM | Homo sapiens | |
19. | ALA1475629 | SID85147440 | AC50 | > | 70 | uM | ALA3214889 | inactive | nM | Homo sapiens | ||
20. | 3-Amino-4-hydroxy-5-nitrobenzenesulfonic Acid | SID24841228 | AC50 | > | 70 | uM | ALA3214889 | inactive | nM | Homo sapiens |