# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4283703 | (+/-)-1 | Activity | 0 | ALA4256544 | Not Active | Rattus norvegicus | |||||
2. | ALA1086654 | 4 | Imax | 0 | ALA4256540 | Not Determined | Rattus norvegicus | |||||
3. | ALA4290888 | (2aR,4aS,9aS)-1 | Imax | 0 | ALA4256540 | Not Determined | Rattus norvegicus | |||||
4. | ALA4283703 | (+/-)-1 | Imax | = | 0.79 | % | ALA4256540 | % | Rattus norvegicus | |||
5. | Acetylcholine | table I | EC50 | 0 | ALA4256539 | Not Determined | Rattus norvegicus | |||||
6. | ALA1086654 | 4 | EC50 | 0 | ALA4256539 | Not Determined | Rattus norvegicus | |||||
7. | ALA4290888 | (2aR,4aS,9aS)-1 | EC50 | 0 | ALA4256539 | Not Determined | Rattus norvegicus | |||||
8. | ALA4283703 | (+/-)-1 | EC50 | = | 29 | uM | ALA4256539 | 4.54 | nM | Rattus norvegicus | ||
9. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033574 | Not Active | Rattus norvegicus | |||||
10. | ALA327197 | 5 | IC50 | = | 0.37 | nM | ALA4844593 | 9.43 | nM | Rattus norvegicus | ||
11. | ALA2204360 | 5m, Lu AA21004 | Ki | = | 230 | nM | ALA2215366 | 6.64 | nM | Rattus norvegicus | ||
12. | ALA2204360 | 5m, Lu AA21004 | IC50 | = | 0.18 | nM | ALA2215819 | 9.74 | nM | Rattus norvegicus | ||
13. | Ondansetron | 2 | IC50 | = | 0.16 | nM | ALA2215819 | 9.80 | nM | Rattus norvegicus | ||
14. | ALA2204360 | 5m, Lu AA21004 | Activity | 0 | ALA2215369 | Not Active | Rattus norvegicus | |||||
15. | ALA2011600 | 6f | Ki | = | 71 | nM | ALA2015860 | 7.15 | nM | Rattus norvegicus | ||
16. | ALA2011599 | 6e | Ki | = | 89 | nM | ALA2015860 | 7.05 | nM | Rattus norvegicus | ||
17. | ALA2011598 | 6d | Ki | = | 132 | nM | ALA2015860 | 6.88 | nM | Rattus norvegicus | ||
18. | ALA2011597 | 6c | Ki | = | 127 | nM | ALA2015860 | 6.90 | nM | Rattus norvegicus | ||
19. | ALA2011596 | 6b | Ki | = | 18 | nM | ALA2015860 | 7.75 | nM | Rattus norvegicus | ||
20. | ALA2011595 | 6a | Ki | = | 178 | nM | ALA2015860 | 6.75 | nM | Rattus norvegicus |