# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5191950 | DT2216 | EC50 | = | 63 | nM | ALA5127824 | 7.20 | nM | Homo sapiens | ||
2. | ALA5186923 | 27; DT-2216 | Emax | = | 26 | % | ALA5124521 | % | Homo sapiens | |||
3. | ALA5186923 | 27; DT-2216 | DC50 | > | 3 | uM | ALA5124520 | uM | Homo sapiens | |||
4. | ALA5186923 | 27; DT-2216 | Emax | = | 91 | % | ALA5124519 | % | Homo sapiens | |||
5. | ALA5186923 | 27; DT-2216 | DC50 | = | 63 | nM | ALA5124518 | nM | Homo sapiens | |||
6. | ALA5205953 | 29 | Emax | = | 76 | % | ALA5108732 | % | Homo sapiens | |||
7. | ALA5205953 | 29 | EC50 | = | 4.8 | nM | ALA5108731 | 8.32 | nM | Homo sapiens | ||
8. | DT2216 | 1e; DT2216 | Emax | = | 90.8 | % | ALA5108725 | % | Homo sapiens | |||
9. | DT2216 | 1e; DT2216 | EC50 | = | 63 | nM | ALA5108724 | 7.20 | nM | Homo sapiens | ||
10. | ALA5197462 | DT2216 | Emax | = | 90.8 | % | ALA5104686 | % | Homo sapiens | |||
11. | ALA5197462 | DT2216 | EC50 | = | 63 | nM | ALA5104685 | 7.20 | nM | Homo sapiens | ||
12. | ALA5092688 | PZ703b-NC | Activity | 0 | ALA5054297 | Not Active | Homo sapiens | |||||
13. | ALA5077514 | PZ703b | Activity | 0 | ALA5054297 | Not Active | Homo sapiens | |||||
14. | ALA5087367 | DT2216 | Activity | 0 | ALA5054297 | Not Active | Homo sapiens | |||||
15. | ALA443684 | Scheme 4, 11 | Activity | 0 | ALA5054297 | Not Active | Homo sapiens | |||||
16. | ALA5092688 | PZ703b-NC | Activity | 0 | ALA5054295 | Active | Homo sapiens | |||||
17. | ALA5077514 | PZ703b | Activity | 0 | ALA5054295 | Active | Homo sapiens | |||||
18. | ALA5087367 | DT2216 | Activity | 0 | ALA5054295 | Active | Homo sapiens | |||||
19. | ALA443684 | Scheme 4, 11 | Activity | 0 | ALA5054295 | Active | Homo sapiens | |||||
20. | ALA5092688 | PZ703b-NC | Activity | 0 | ALA5054292 | Not Active | Homo sapiens |