# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4446933 | 6 | IC50 | = | 2.8 | uM | ALA4415948 | 5.55 | nM | Homo sapiens | ||
2. | ALA4444045 | 3 | IC50 | = | 2.8 | uM | ALA4415948 | 5.55 | nM | Homo sapiens | ||
3. | ALA4452883 | 2 | IC50 | = | 2.8 | uM | ALA4415948 | 5.55 | nM | Homo sapiens | ||
4. | ALA4452781 | 1 | IC50 | = | 2.8 | uM | ALA4415948 | 5.55 | nM | Homo sapiens | ||
5. | N-(4-{3-[2-(methylcarbamoyl)ethyl]-5-[4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl]-1H-pyrazol-1-yl}phenyl)prop-2-ynamide | 1; Tr-87 | Activity | 0 | ALA4415379 | Active | Homo sapiens | |||||
6. | (-)-Hydroxycitric acid | 3 | Ki | = | 0.3 | mM | ALA4275769 | nM | Homo sapiens | |||
7. | ALA2165262 | 126-(-) | Ki | = | 0.7 | uM | ALA4275769 | 6.16 | nM | Homo sapiens | ||
8. | ALA2165261 | 125-(+) | Ki | = | 3.2 | uM | ALA4275769 | 5.50 | nM | Homo sapiens | ||
9. | ALA1214277 | 1 | IC50 | = | 7 | uM | ALA4275770 | 5.16 | nM | Homo sapiens | ||
10. | Radicicol | 1 (radicicol) | INH | = | 50 | % | ALA4275774 | % | Homo sapiens | |||
11. | ALA119628 | 45 | Ki | = | 1 | uM | ALA4275779 | 6.00 | nM | Homo sapiens | ||
12. | ALA120302 | 76 | Ki | = | 220 | nM | ALA4275779 | 6.66 | nM | Homo sapiens | ||
13. | SB 204990 | (-)-77 | INH | = | 91 | % | ALA4275780 | % | Homo sapiens | |||
14. | SB 204990 | (-)-77 | INH | = | 82 | % | ALA4275781 | % | Homo sapiens | |||
15. | (-)-Hydroxycitric acid | 3 | INH | 0 | ALA4001976 | Active | % | Homo sapiens | ||||
16. | ALA119628 | 45 | INH | 0 | ALA4001976 | Active | % | Homo sapiens | ||||
17. | ALA4061755 | C4 | Activity | = | 58.8 | % | ALA4001975 | % | Homo sapiens | |||
18. | ALA4061755 | C4 | Activity | = | 31.4 | % | ALA4001974 | % | Homo sapiens | |||
19. | ALA4061755 | C4 | Activity | = | 81.2 | % | ALA4001973 | % | Homo sapiens | |||
20. | ALA4061755 | C4 | Activity | = | 11.9 | % | ALA4001972 | % | Homo sapiens |