| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  BI-3812 | 44 | % Ctrl | = | 101 | % | ALA5304288 | Not Active | % | Homo sapiens | ||
| 2. |  BI-3802 | BI-3802 | % Ctrl | = | 90 | % | ALA5304185 | Not Active | % | Homo sapiens | ||
| 3. |  ALA3774448 | 17 | IC50 | = | 157 | nM | ALA3776317 | 6.80 | nM | Homo sapiens | ||
| 4. | ALA3774448 | 17 | INH | = | 35 | % | ALA3776501 | % | Homo sapiens | |||
| 5. |  ALA3775393 | 16 | INH | 0 | ALA3776320 | Not Active | % | Homo sapiens | ||||
| 6. | ALA3774448 | 17 | INH | = | 89 | % | ALA3776316 | % | Homo sapiens | |||
| 7. | ALA3775393 | 16 | INH | = | 12 | % | ALA3776315 | % | Homo sapiens | |||
| 8. |  ALA3758502 | 1 | INH | = | -15.9 | % | ALA3760653 | % | Homo sapiens | |||
| 9. |  ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3748000 | nM | Homo sapiens | |||
| 10. |  ALA3628628 | 5 | INH | = | 12.11 | % | ALA3631445 | % | Homo sapiens | |||
| 11. |  ALA3628627 | 4 | INH | = | 30.2 | % | ALA3631445 | % | Homo sapiens | |||
| 12. |  ALA166031 | 3 | INH | = | 53.19 | % | ALA3631445 | % | Homo sapiens | |||
| 13. |  SGC AAK1 1 | 25; SGC-AAK1-1 | Kd | = | 960 | nM | ALA5213596 | 6.02 | nM | Homo sapiens | ||
| 14. |  ALA5199698 | 58 | IC50 | = | 0.45 | uM | ALA5161246 | 6.35 | nM | Homo sapiens | ||
| 15. |  ALA4092824 | 122 | IC50 | = | 0.35 | uM | ALA5161246 | 6.46 | nM | Homo sapiens | ||
| 16. |  ALA5195653 | 46 | IC50 | = | 0.6 | uM | ALA5161246 | 6.22 | nM | Homo sapiens | ||
| 17. |  ALA5205578 | 44 | IC50 | = | 0.65 | uM | ALA5161246 | 6.19 | nM | Homo sapiens | ||
| 18. |  ALA5170576 | 43 | IC50 | = | 1.8 | uM | ALA5161246 | 5.75 | nM | Homo sapiens | ||
| 19. |  ALA5179796 | b27 | INH | 0 | ALA5144373 | NA | % | Homo sapiens | ||||
| 20. |  ALA5179350 | b23 | INH | = | 18 | % | ALA5144372 | % | Homo sapiens |
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