# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288241 | B2 | INH | < | 50 | % | ALA5238264 | % | Homo sapiens | |||
2. | Defactinib | DEFACTINIB | IC50 | = | 75.3 | nM | ALA5213450 | 7.12 | nM | Homo sapiens | ||
3. | 4-(6-((4-Ethynylpyrimidin-2-yl)Ethynyl)-1H-Benzo[d]Imidazol-1-yl)Pyrimidin-2-Amine | 18 | INH | > | 50 | % | ALA5151677 | % | Homo sapiens | |||
4. | ALA5183704 | 22 | INH | = | 7 | % | ALA5119685 | % | Homo sapiens | |||
5. | ALA4463436 | 28 | INH | = | 96 | % | ALA4429534 | % | Homo sapiens | |||
6. | ALA4463436 | 28 | INH | = | 84 | % | ALA4429553 | % | Homo sapiens | |||
7. | ALA4463436 | 28 | INH | = | 26 | % | ALA4429556 | % | Homo sapiens | |||
8. | ALA4564126 | 18 | INH | <= | 16 | % | ALA4427660 | % | Homo sapiens | |||
9. | ALA4564126 | 18 | IC50 | >= | 5 | uM | ALA4427716 | nM | Homo sapiens | |||
10. | ALA4445335 | Roxyl-ZV-5J | INH | = | 1 | % | ALA4408048 | % | Homo sapiens | |||
11. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405458 | % | Homo sapiens | |||
12. | ALA4555782 | 24 | Activity | = | 24 | % | ALA4400068 | % | Homo sapiens | |||
13. | ALA4559936 | (+/-)-6 | Activity | = | 38 | % | ALA4391449 | % | Homo sapiens | |||
14. | ALA4564973 | 50 | INH | = | 86 | % | ALA4389823 | % | Homo sapiens | |||
15. | ALA4555459 | 43 | INH | = | 59 | % | ALA4389346 | % | Homo sapiens | |||
16. | ALA4545456 | 24 | INH | = | 47 | % | ALA4387295 | % | Homo sapiens | |||
17. | Abemaciclib | ABEMACICLIB | INH | = | 11.5 | % | ALA4387295 | % | Homo sapiens | |||
18. | ALA4473365 | 7c | Activity | = | 39 | % | ALA4382627 | % | Homo sapiens | |||
19. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379257 | nM | Homo sapiens | |||
20. | ALA4459587 | DC-TEADin02 | INH | = | 8 | % | ALA4378943 | % | Homo sapiens |