# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4848198 | UM208 | IC50 | = | 2.11 | 10^-6M | ALA4807524 | 5.68 | nM | Rattus norvegicus | ||
2. | ALA4852279 | UM207 | IC50 | = | 1.52 | 10^-8M | ALA4807524 | 7.82 | nM | Rattus norvegicus | ||
3. | ALA4849630 | UM206 | IC50 | = | 1.69 | 10^-11M | ALA4807524 | 10.77 | nM | Rattus norvegicus | ||
4. | ALA4861317 | Table 1, R22C1 | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
5. | ALA4849595 | UM206 (4 T = A, 7 G = A, 9 D = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
6. | ALA4872198 | UM206 ( 12-13 EL=AA) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
7. | ALA4855070 | UM206 (13 L = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
8. | ALA4864995 | UM206 (12 E = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
9. | ALA4877748 | UM206 (11 C = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
10. | ALA4859312 | UM206 (10 G = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
11. | ALA4860112 | UM206 (9 D = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
12. | ALA4870480 | UM206 (8 M = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
13. | ALA4850145 | UM206 (7 G = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
14. | ALA4871325 | UM206 (6 E = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
15. | ALA4847646 | UM206 (5 S = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
16. | ALA4861360 | UM206 (4 T = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
17. | ALA4847975 | UM206 (3 K = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
18. | ALA4854336 | UM206 (2 N = A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
19. | ALA4847233 | UM206 (1 C= A) | INH | 0 | ALA4807455 | Not Active | % | Rattus norvegicus | ||||
20. | ALA4861317 | Table 1, R22C1 | INH | 0 | ALA4807453 | Not Active | % | Rattus norvegicus |