# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5206366 | 13; JNJ-64264681 | Activity | 0 | ALA5152699 | Dde | Rattus norvegicus | |||||
2. | ALA4877846 | 30 | IC50 | = | 11 | nM | ALA4822497 | 7.96 | nM | Rattus norvegicus | ||
3. | rilzabrutinib | BDBM143212 | Activity | = | 95 | % | ALA5104989 | % | Rattus norvegicus | |||
4. | rilzabrutinib | BDBM143212 | Activity | = | 98 | % | ALA5104988 | % | Rattus norvegicus | |||
5. | rilzabrutinib | BDBM143212 | Activity | = | 95 | % | ALA5104987 | % | Rattus norvegicus | |||
6. | rilzabrutinib | BDBM143212 | Activity | = | 70 | % | ALA5104986 | % | Rattus norvegicus | |||
7. | rilzabrutinib | BDBM143212 | Activity | 0 | ALA5104985 | Dde | Rattus norvegicus | |||||
8. | rilzabrutinib | BDBM143212 | Activity | 0 | ALA5104984 | Dde | Rattus norvegicus | |||||
9. | rilzabrutinib | BDBM143212 | Activity | = | 29 | % | ALA5104979 | % | Rattus norvegicus | |||
10. | rilzabrutinib | BDBM143212 | Activity | = | 80 | % | ALA5104978 | % | Rattus norvegicus | |||
11. | rilzabrutinib | BDBM143212 | Activity | = | 91 | % | ALA5104977 | % | Rattus norvegicus | |||
12. | rilzabrutinib | BDBM143212 | Activity | = | 95 | % | ALA5104976 | % | Rattus norvegicus | |||
13. | atuzabrutinib | BDBM197260 | Activity | = | 81.9 | % | ALA5104954 | % | Rattus norvegicus | |||
14. | atuzabrutinib | BDBM197260 | Activity | = | 48.7 | % | ALA5104953 | % | Rattus norvegicus | |||
15. | atuzabrutinib | BDBM197260 | Activity | = | 36.3 | % | ALA5104952 | % | Rattus norvegicus | |||
16. | atuzabrutinib | BDBM197260 | Activity | = | 87.3 | % | ALA5104948 | % | Rattus norvegicus | |||
17. | atuzabrutinib | BDBM197260 | Activity | = | 50.1 | % | ALA5104947 | % | Rattus norvegicus | |||
18. | atuzabrutinib | BDBM197260 | Activity | = | 33.9 | % | ALA5104946 | % | Rattus norvegicus |