# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Raloxifene | 44 | IC50 | = | 5.7 | nM | ALA5233653 | 8.24 | nM | Homo sapiens | ||
2. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | IC50 | = | 5 | nM | ALA5233652 | 8.30 | nM | Homo sapiens | ||
3. | β-Estradiol | Table II | IC50 | = | 5 | nM | ALA5233652 | 8.30 | nM | Homo sapiens | ||
4. | Genistein | 1 (Genistein) | IC50 | = | 5 | nM | ALA5233652 | 8.30 | nM | Homo sapiens | ||
5. | Perphenazine | perphenazine | IC50 | < | 1 | uM | ALA5233652 | nM | Homo sapiens | |||
6. | Chlorpromazine | cholrpromazine | IC50 | < | 1 | uM | ALA5233652 | nM | Homo sapiens | |||
7. | FXIa inhibitor 3f | 3f | t1/2 | > | 180 | min | ALA5141415 | hr | Homo sapiens | |||
8. | Raloxifene | 44 | IC50 | = | 0.045 | uM | ALA4420028 | 7.35 | nM | Homo sapiens | ||
9. | Menadione | Menadione | IC50 | = | 99.2 | uM | ALA4420028 | 4.00 | nM | Homo sapiens | ||
10. | Tamoxifen | Tamoxifen | IC50 | = | 97.3 | uM | ALA4420028 | 4.01 | nM | Homo sapiens | ||
11. | ALA42 | clozapine | IC50 | = | 43.3 | uM | ALA4420028 | 4.36 | nM | Homo sapiens | ||
12. | ALA532 | Ery | IC50 | = | 96.9 | uM | ALA4420028 | 4.01 | nM | Homo sapiens | ||
13. | Hydralazine | Hydralazyne | IC50 | = | 3.93 | uM | ALA4420028 | 5.41 | nM | Homo sapiens | ||
14. | Dehydroepiandrosterone sulfate | Dehydroepiandrosterone sulfate (DHEAS) | IC50 | > | 100 | uM | ALA4420028 | nM | Homo sapiens | |||
15. | ALA4575293 | 11a | Activity | 0 | ALA4416705 | Not Active | Homo sapiens | |||||
16. | AZD7648 | Example 16; AZD7648 | Drug metabolism | 0 | ALA4403963 | Metabolite_Notdetected | Homo sapiens | |||||
17. | AZD7648 | Example 16; AZD7648 | Drug metabolism | 0 | ALA4403962 | Metabolite_Notdetected | Homo sapiens | |||||
18. | GSK2983559 active metabolite | 5 | Activity | 0 | ALA4367456 | Not Active | Homo sapiens | |||||
19. | GSK2983559 active metabolite | 5 | Activity | 0 | ALA4367455 | Not Active | Homo sapiens | |||||
20. | ALA4587320 | M1 | Drug uptake | 0 | ALA4326440 | Active | Homo sapiens |