# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5189893 | 19; VU6015241 | IC50 | > | 10000 | nM | ALA5133245 | nM | Rattus norvegicus | |||
2. | ALA295388 | 4j | pKi | = | 9.5 | ALA4397787 | 9.50 | nM | Rattus norvegicus | |||
3. | ALA271108 | 3 | Ki | = | 9 | nM | ALA4183541 | 8.05 | nM | Rattus norvegicus | ||
4. | Tolterodine L-tartrate | Tolterodine | Ki | = | 2.7 | nM | ALA4183541 | 8.57 | nM | Rattus norvegicus | ||
5. | ALA4745892 | Cyclostellettamine A | IC50 | = | 0.026 | mg/ml | ALA4676978 | ug.mL-1 | Rattus norvegicus | |||
6. | ALA4788850 | Cyclostellettamine B | IC50 | = | 0.031 | mg/ml | ALA4676978 | ug.mL-1 | Rattus norvegicus | |||
7. | ALA4743200 | Cyclostellettamine C | IC50 | = | 0.054 | mg/ml | ALA4676978 | ug.mL-1 | Rattus norvegicus | |||
8. | ALA4749898 | Cyclostellettamine D | IC50 | = | 0.059 | mg/ml | ALA4676978 | ug.mL-1 | Rattus norvegicus | |||
9. | ALA4750886 | Cyclostellettamine E | IC50 | = | 0.133 | mg/ml | ALA4676978 | ug.mL-1 | Rattus norvegicus | |||
10. | ALA4797832 | Cyclostellettamine F | IC50 | = | 0.15 | mg/ml | ALA4676978 | ug.mL-1 | Rattus norvegicus | |||
11. | ALA4639776 | 9 | FC | = | 1.6 | ALA4623757 | Rattus norvegicus | |||||
12. | ALA4644670 | 8a; 4b | Ki | = | 7.6 | nM | ALA4605252 | 8.12 | nM | Rattus norvegicus | ||
13. | 4-Piperidyl n-(2-biphenyl)carbamate | 8a | Ki | = | 270 | nM | ALA4605252 | 6.57 | nM | Rattus norvegicus | ||
14. | ML380 | 8n | EC50 | > | 30 | uM | ALA3370309 | nM | Rattus norvegicus | |||
15. | ALA3298763 | 46 | Ki | = | 0.64 | nM | ALA3369302 | 9.19 | nM | Rattus norvegicus | ||
16. | ALA3298601 | 45 | Ki | = | 14 | nM | ALA3369302 | 7.85 | nM | Rattus norvegicus | ||
17. | ALA3298600 | 44 | Ki | = | 0.21 | nM | ALA3369302 | 9.68 | nM | Rattus norvegicus | ||
18. | ALA3298599 | 43 | Ki | = | 0.053 | nM | ALA3369302 | 10.28 | nM | Rattus norvegicus | ||
19. | ALA3298598 | 42 | Ki | = | 1.2 | nM | ALA3369302 | 8.92 | nM | Rattus norvegicus | ||
20. | ALA3298597 | 41 | Ki | = | 1.2 | nM | ALA3369302 | 8.92 | nM | Rattus norvegicus |