# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF-06873600 | PF-06873600 | Ki | < | 0.019 | uM | ALA5244059 | nM | Homo sapiens | |||
2. | Dinaciclib (SCH727965) | DINACICLIB | Ki | = | 0.004 | uM | ALA5244059 | 8.40 | nM | Homo sapiens | ||
3. | ALA5195030 | 4; CYC065 | Ki | = | 0.026 | uM | ALA5244059 | 7.58 | nM | Homo sapiens | ||
4. | AT7519 | 33 | Ki | < | 0.01 | uM | ALA5244059 | nM | Homo sapiens | |||
5. | ALA1782169 | 7a | IC50 | = | 0.24 | uM | ALA5227480 | 6.62 | nM | Homo sapiens | ||
6. | ALA1782170 | 7b | IC50 | = | 7.4 | uM | ALA5227480 | 5.13 | nM | Homo sapiens | ||
7. | ALA1782168 | 6 | IC50 | = | 0.22 | uM | ALA5227480 | 6.66 | nM | Homo sapiens | ||
8. | Kenpaullone | 28a | IC50 | = | 0.064 | uM | ALA5227480 | 7.19 | nM | Homo sapiens | ||
9. | ALA215205 | 31b, (CAN508) | IC50 | = | 350 | nM | ALA5224469 | 6.46 | nM | Homo sapiens | ||
10. | ALA5202522 | 46; MC180295 | IC50 | = | 5 | nM | ALA5224425 | 8.30 | nM | Homo sapiens | ||
11. | ALA5287128 | BAY 1000394 | IC50 | = | 5 | nM | ALA5224425 | 8.30 | nM | Homo sapiens | ||
12. | ALA5283615 | Table1, R11C5 | IC50 | = | 9 | nM | ALA5253276 | 8.05 | nM | Homo sapiens | ||
13. | ALA5283233 | Table1, R10C5 | IC50 | = | 7 | nM | ALA5253276 | 8.15 | nM | Homo sapiens | ||
14. | ALA5272545 | Table1, R9C5 | IC50 | = | 6 | nM | ALA5253276 | 8.22 | nM | Homo sapiens | ||
15. | ALA5288282 | Table1, R8C5 | IC50 | = | 8 | nM | ALA5253276 | 8.10 | nM | Homo sapiens | ||
16. | ALA5290495 | Table1, R7C5 | IC50 | = | 7 | nM | ALA5253276 | 8.15 | nM | Homo sapiens |