# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Estriol | 4 | RBA | = | 21 | % | ALA3136672 | % | Rattus norvegicus | |||
2. | ALA1950809 | 2, S-DPN | Ki | = | 1.82 | nM | ALA1954168 | 8.74 | nM | Rattus norvegicus | ||
3. | (R)-DPN | DPN(1)(table 1) | Ki | = | 0.27 | nM | ALA1954168 | 9.57 | nM | Rattus norvegicus | ||
4. | ALA469316 | 41d | IC50 | = | 14.2 | uM | ALA940318 | 4.85 | nM | Rattus norvegicus | ||
5. | ALA472469 | 36c | IC50 | = | 828 | nM | ALA940318 | 6.08 | nM | Rattus norvegicus | ||
6. | ALA371012 | 14 | Activity | = | 78 | % | ALA870538 | % | Rattus norvegicus | |||
7. | ALA371012 | 14 | EC50 | = | 1.09 | nM | ALA868727 | 8.96 | nM | Rattus norvegicus | ||
8. | ALA200799 | 11 | Activity | = | 93 | % | ALA870538 | % | Rattus norvegicus | |||
9. | ALA200799 | 11 | EC50 | = | 6.7 | nM | ALA868727 | 8.17 | nM | Rattus norvegicus | ||
10. | ALA199599 | 7c | Activity | = | 101 | % | ALA870538 | % | Rattus norvegicus | |||
11. | ALA199599 | 7c | EC50 | = | 40.8 | nM | ALA868727 | 7.39 | nM | Rattus norvegicus | ||
12. | β-Estradiol | Table II | Activity | = | 100 | % | ALA870538 | % | Rattus norvegicus | |||
13. | β-Estradiol | Table II | EC50 | = | 0.14 | nM | ALA868727 | 9.85 | nM | Rattus norvegicus | ||
14. | ALA537638 | 17 | Ki | = | 0.3 | nM | ALA884932 | 9.52 | nM | Rattus norvegicus | ||
15. | ALA536733 | 16 | Ki | = | 1.36 | nM | ALA884932 | 8.87 | nM | Rattus norvegicus | ||
16. | ALA557981 | 9 | Ki | = | 24.1 | nM | ALA884932 | 7.62 | nM | Rattus norvegicus | ||
17. | ALA539849 | 2 | Ki | = | 0.7 | nM | ALA884932 | 9.15 | nM | Rattus norvegicus | ||
18. | Raloxifene HCl | 50 | Ki | = | 2.74 | nM | ALA884932 | 8.56 | nM | Rattus norvegicus | ||
19. | β-Estradiol | Table II | IC50 | = | 1.7 | nM | ALA828749 | 8.77 | nM | Rattus norvegicus | ||
20. | ALA188882 | 36 | IC50 | = | 36 | nM | ALA828749 | 7.44 | nM | Rattus norvegicus |