# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3126388 | Dec-RVKR-CMK | Ki | = | 3.6 | nM | ALA4428332 | 8.44 | nM | Homo sapiens | ||
2. | ALA2179430 | hPC7, Q16549 | Ki | = | 0.34 | nM | ALA2187699 | 9.47 | nM | Homo sapiens | ||
3. | ALA2179835 | hfurin, P09958 | Ki | = | 0.4 | nM | ALA2187699 | 9.40 | nM | Homo sapiens | ||
4. | ALA2179836 | mPC1/3, P63239 | Ki | = | 1.1 | nM | ALA2187699 | 8.96 | nM | Homo sapiens | ||
5. | ALA2179429 | hPC5/6, Q92824 | Ki | = | 1.3 | nM | ALA2187699 | 8.89 | nM | Homo sapiens | ||
6. | ALA2179431 | hPACE4, P29122 | Ki | = | 2 | nM | ALA2187699 | 8.70 | nM | Homo sapiens | ||
7. | ALA2179428 | mPC4, P2921 | Ki | = | 7 | nM | ALA2187699 | 8.15 | nM | Homo sapiens | ||
8. | ALA2179434 | Ac-LLLRVKR-NH2 | Ki | = | 18 | nM | ALA2187699 | 7.75 | nM | Homo sapiens | ||
9. | ALA2179832 | Ac-[PEG8]LLLLRVKR-NH2 | Ki | = | 19 | nM | ALA2187699 | 7.72 | nM | Homo sapiens | ||
10. | ALA2179435 | Ac-LLLLRVKR-NH2 | Ki | = | 22 | nM | ALA2187699 | 7.66 | nM | Homo sapiens | ||
11. | ALA2179833 | Ac-[C8]LLLLRVKR-NH2 | Ki | = | 23 | nM | ALA2187699 | 7.64 | nM | Homo sapiens | ||
12. | ALA2179436 | Ac-LLLLLRVKR-NH2 | Ki | = | 70 | nM | ALA2187699 | 7.16 | nM | Homo sapiens | ||
13. | ALA2049156 | 17 | Ki | = | 240 | nM | ALA2187699 | 6.62 | nM | Homo sapiens | ||
14. | ALA2179437 | Ac-LLLLLLRVKR-NH2 | Ki | = | 300 | nM | ALA2187699 | 6.52 | nM | Homo sapiens | ||
15. | ALA2179427 | hPC2, P16519 | Ki | > | 1000 | nM | ALA2187699 | nM | Homo sapiens | |||
16. | ALA2179432 | Ac-RVKR-NH2 | Ki | = | 1600 | nM | ALA2187699 | 5.80 | nM | Homo sapiens | ||
17. | ALA2179433 | Ac-LRVKR-NH2 | Ki | = | 1600 | nM | ALA2187699 | 5.80 | nM | Homo sapiens | ||
18. | ALA2179438 | Ac-LLLLRVK[DArg]-NH2 | Ki | = | 1380 | nM | ALA2187699 | 5.86 | nM | Homo sapiens | ||
19. | ALA4785628 | CF12 | INH | 0 | ALA4689551 | Active | % | Homo sapiens | ||||
20. | ALA4793978 | CF8 | INH | 0 | ALA4689551 | Active | % | Homo sapiens |