# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 2 | uM | ALA5252876 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 2 | uM | ALA5252876 | nM | Homo sapiens | |||
3. | ALA5273533 | 37 | IC50 | > | 1000 | nM | ALA5244429 | nM | Homo sapiens | |||
4. | ALA5281283 | 18 | IC50 | > | 1000 | nM | ALA5244429 | nM | Homo sapiens | |||
5. | ALA3701197 | BDBM161028 | % of control | = | 38 | % | ALA5214566 | % | Homo sapiens | |||
6. | ALA5185626 | 83 | IC50 | > | 49.5 | uM | ALA5140655 | nM | Homo sapiens | |||
7. | ALA4466696 | 32 | pIC50 | = | 7 | ALA4433071 | 7.00 | nM | Homo sapiens | |||
8. | ALA4463436 | 28 | INH | = | -2 | % | ALA4429548 | % | Homo sapiens | |||
9. | JTE-952 | JTE-952; (S)-8b | IC50 | > | 1000 | nM | ALA4424915 | nM | Homo sapiens | |||
10. | ALA4445335 | Roxyl-ZV-5J | INH | = | 11 | % | ALA4408175 | % | Homo sapiens | |||
11. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405622 | % | Homo sapiens | |||
12. | ALA4559936 | (+/-)-6 | Activity | = | 60 | % | ALA4391649 | % | Homo sapiens | |||
13. | ALA4564973 | 50 | INH | = | 80 | % | ALA4390023 | % | Homo sapiens | |||
14. | ALA4555459 | 43 | INH | = | 75 | % | ALA4389546 | % | Homo sapiens | |||
15. | ALA4545456 | 24 | INH | = | 7 | % | ALA4387382 | % | Homo sapiens | |||
16. | Abemaciclib | ABEMACICLIB | INH | = | -0.5 | % | ALA4387382 | % | Homo sapiens | |||
17. | ALA4473365 | 7c | Activity | = | 77 | % | ALA4382827 | % | Homo sapiens | |||
18. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379493 | nM | Homo sapiens | |||
19. | ALA4459587 | DC-TEADin02 | INH | = | 5 | % | ALA4378986 | % | Homo sapiens | |||
20. | CDK9-IN-7 | 21e | INH | = | 13 | % | ALA4377982 | % | Homo sapiens |