# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Canertinib (CI-1033) | 18 | IC50 | = | 0.12 | uM | ALA5236037 | 6.92 | nM | Homo sapiens | ||
2. | ALA5269225 | 28; GSK2793660 | IC50 | = | 1 | nM | ALA5236037 | 9.00 | nM | Homo sapiens | ||
3. | ALA1192402 | 34 | IC50 | = | 39 | uM | ALA5236036 | 4.41 | nM | Homo sapiens | ||
4. | IcatCXPZ₋₀₁ | IcatCXPZ-01 | IC5 | = | 15 | nM | ALA5236035 | nM | Homo sapiens | |||
5. | ALA1242565 | 2, JCP405 | Ratio | = | 2 | 10^6/M/s | ALA5236034 | 10^6/M/s | Homo sapiens | |||
6. | ALA5290773 | 6 | Ratio | = | 2900 | /M/s | ALA5236034 | /M/s | Homo sapiens | |||
7. | ALA450997 | Gly-4-(I)Phe-DMK | IC50 | = | 1 | nM | ALA5236033 | 9.00 | nM | Homo sapiens | ||
8. | ALA448143 | Gly-Phe-DMK | IC50 | = | 50 | nM | ALA5236033 | 7.30 | nM | Homo sapiens | ||
9. | ALA1242565 | 2, JCP405 | ID50 | = | 0.1 | uM | ALA5236029 | uM | Homo sapiens | |||
10. | ALA5290773 | 6 | IC50 | = | 4.9 | uM | ALA5236029 | 5.31 | nM | Homo sapiens | ||
11. | ALA448143 | Gly-Phe-DMK | INH | > | 90 | % | ALA5236029 | % | Homo sapiens | |||
12. | ALA5186557 | SF38 | Activity | 0 | ALA5165070 | Active | Homo sapiens | |||||
13. | ALA5186557 | SF38 | Activity | 0 | ALA5165034 | Active | Homo sapiens | |||||
14. | ALA5179212 | SF26 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens | |||
15. | ALA5175900 | SF21 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens | |||
16. | ALA5173569 | SF20 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens | |||
17. | ALA5191730 | SF18 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens | |||
18. | ALA5186113 | SF17 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens | |||
19. | ALA5198107 | SF16 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens | |||
20. | ALA5176578 | SF15 | IC50 | > | 5000 | nM | ALA5165029 | nM | Homo sapiens |