# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | DMP696 | 37 DMP-696 | Ki | = | 1.7 | nM | ALA5242047 | 8.77 | nM | Homo sapiens | ||
2. | ALA5269179 | Cpd C | IC50 | = | 16.3 | nM | ALA5237511 | 7.79 | nM | Homo sapiens | ||
3. | ALA5280146 | Cpd B | IC50 | = | 120 | nM | ALA5237511 | 6.92 | nM | Homo sapiens | ||
4. | ALA498311 | MTIP | Ki | = | 9.98 | nM | ALA5237509 | 8.00 | nM | Homo sapiens | ||
5. | ALA121896 | 18n | IC50 | = | 76 | nM | ALA5121348 | 7.12 | nM | Homo sapiens | ||
6. | ALA65078 | 10j | IC50 | = | 76 | nM | ALA5121348 | 7.12 | nM | Homo sapiens | ||
7. | ALA4793451 | 4j; MGS0274 | Activity | 0 | ALA4708763 | Not Active | Homo sapiens | |||||
8. | ALA334014 | 3 | Activity | 0 | ALA4708763 | Not Active | Homo sapiens | |||||
9. | Belzutifan | 2; PT2977 | Activity | 0 | ALA4312721 | Not Active | Homo sapiens | |||||
10. | CHDI 00390576 | 22 | INH | < | 25 | % | ALA4311074 | % | Homo sapiens | |||
11. | ALA4437833 | 16 | INH | < | 25 | % | ALA4311074 | % | Homo sapiens | |||
12. | ALA3793277 | 29k | IC50 | = | 9.5 | nM | ALA4221048 | 8.02 | nM | Homo sapiens | ||
13. | ALA4228089 | (S)-42c | IC50 | = | 350 | nM | ALA4221048 | 6.46 | nM | Homo sapiens | ||
14. | ALA4225709 | (R)-42c | IC50 | = | 58 | nM | ALA4221048 | 7.24 | nM | Homo sapiens | ||
15. | ALA4224781 | 42e | IC50 | = | 46 | nM | ALA4221048 | 7.34 | nM | Homo sapiens | ||
16. | ALA4227282 | 42d | IC50 | = | 100 | nM | ALA4221048 | 7.00 | nM | Homo sapiens | ||
17. | ALA4225039 | 42h | IC50 | = | 210 | nM | ALA4221048 | 6.68 | nM | Homo sapiens | ||
18. | ALA4227177 | 42g | IC50 | = | 320 | nM | ALA4221048 | 6.50 | nM | Homo sapiens | ||
19. | ALA4226158 | 42c | IC50 | = | 110 | nM | ALA4221048 | 6.96 | nM | Homo sapiens | ||
20. | ALA4225373 | 42b | IC50 | = | 48 | nM | ALA4221048 | 7.32 | nM | Homo sapiens |