# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | N-(4-Chloro-3-(trifluoromethyl)phenyl)-4-(6-(4-(4-methylpiperazin-1-yl)phenyl)thieno[2,3-d]pyrimidin-4-yl)piperazine-1-carboxamide | 38k | Activity | 0 | ALA4839217 | Not Active | Mus musculus | |||||
2. | ALA2037208 | 4 | IC50 | = | 2.2 | uM | ALA2038872 | 5.66 | nM | Mus musculus | ||
3. | ALA2037209 | 5 | IC50 | > | 10 | uM | ALA2038872 | nM | Mus musculus | |||
4. | ALA2037211 | 7 | IC50 | = | 3.6 | uM | ALA2038872 | 5.44 | nM | Mus musculus | ||
5. | ALA2037220 | 16 | IC50 | = | 3.2 | uM | ALA2038872 | 5.50 | nM | Mus musculus | ||
6. | ALA2037224 | 20 | IC50 | = | 1.5 | uM | ALA2038872 | 5.82 | nM | Mus musculus | ||
7. | GNF 5837 | 22, GNF-5837 | IC50 | = | 4.4 | uM | ALA2038872 | 5.36 | nM | Mus musculus | ||
8. | SU4312 | 1 | IC50 | = | 0.8 | uM | ALA818398 | 6.10 | nM | Mus musculus | ||
9. | ALA330321 | 52 | IC50 | = | 1 | uM | ALA818398 | 6.00 | nM | Mus musculus | ||
10. | ALA88405 | 18 | IC50 | > | 50 | uM | ALA818398 | nM | Mus musculus | |||
11. | SU 4984 | 16 | IC50 | = | 1.6 | uM | ALA818398 | 5.80 | nM | Mus musculus | ||
12. | ALA86921 | 13 | IC50 | = | 22.6 | uM | ALA818398 | 4.65 | nM | Mus musculus | ||
13. | ALA89721 | 56 | IC50 | = | 2.34 | uM | ALA818398 | 5.63 | nM | Mus musculus | ||
14. | ALA86944 | 36 | IC50 | > | 100 | uM | ALA818398 | nM | Mus musculus | |||
15. | ALA89505 | 29 | IC50 | = | 8.4 | uM | ALA818398 | 5.08 | nM | Mus musculus | ||
16. | Semaxanib (SU5416) | 5a | IC50 | = | 1.04 | uM | ALA818398 | 5.98 | nM | Mus musculus | ||
17. | 3-(4-Isopropylbenzylidenyl)indolin-2-one | Table 1 | IC50 | = | 5.2 | uM | ALA818398 | 5.28 | nM | Mus musculus | ||
18. | ALA89646 | 63 | IC50 | > | 100 | uM | ALA818398 | nM | Mus musculus | |||
19. | ALA89809 | 14 | IC50 | = | 3 | uM | ALA818398 | 5.52 | nM | Mus musculus | ||
20. | ALA87810 | 26 | IC50 | = | 7.6 | uM | ALA818398 | 5.12 | nM | Mus musculus |