# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4574669 | (R,R)-36n | INH | 0 | ALA4351920 | Not Active | % | Mus musculus | ||||
2. | ALA4472294 | 11g | Activity | = | 3 | % | ALA4336969 | % | Mus musculus | |||
3. | ALA4207014 | 19 | INH | = | 45 | % | ALA4191031 | % | Mus musculus | |||
4. | TC-S 7001 | SID103905649 | % inhibition | 4 | % | ALA4881533 | Not Active | % | Mus musculus | |||
5. | Plinabulin (NPI-2358) | 1, NPI-2358/KPU-2 | INH | > | 50 | % | ALA3881642 | % | Mus musculus | |||
6. | Plinabulin (NPI-2358) | 1, NPI-2358/KPU-2 | IC50 | = | 11.1 | uM | ALA3881646 | 4.96 | nM | Mus musculus | ||
7. | ALA2037208 | 4 | IC50 | = | 7.1 | uM | ALA2038984 | 5.15 | nM | Mus musculus | ||
8. | ALA2037209 | 5 | IC50 | = | 6.6 | uM | ALA2038984 | 5.18 | nM | Mus musculus | ||
9. | ALA2037211 | 7 | IC50 | = | 6 | uM | ALA2038984 | 5.22 | nM | Mus musculus | ||
10. | ALA2037220 | 16 | IC50 | > | 10 | uM | ALA2038984 | nM | Mus musculus | |||
11. | ALA2037224 | 20 | IC50 | = | 1.9 | uM | ALA2038984 | 5.72 | nM | Mus musculus | ||
12. | GNF 5837 | 22, GNF-5837 | IC50 | = | 7.3 | uM | ALA2038984 | 5.14 | nM | Mus musculus | ||
13. | ALA1644616 | 1 | INH | = | 100 | % | ALA1646184 | % | Mus musculus | |||
14. | MLN8054 | MLN-8054 | Activity | = | 52 | % | ALA921984 | % | Mus musculus | |||
15. | ALA397771 | 9b | Inhibition | = | 99 | % | ALA886982 | % | Mus musculus | |||
16. | ALA396327 | 10b | Inhibition | = | 104 | % | ALA886982 | % | Mus musculus | |||
17. | ALA1162963 | 3 | Inhibition | = | 90 | % | ALA886982 | % | Mus musculus | |||
18. | ALA247067 | 9a | Inhibition | = | 102 | % | ALA886982 | % | Mus musculus | |||
19. | ALA109981 | 14 | Activity | = | 20 | % | ALA769209 | % | Mus musculus | |||
20. | ALA109944 | 9f | Activity | = | 81 | % | ALA769209 | % | Mus musculus |