| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5189893 | 19; VU6015241 | IC50 | > | 10000 | nM | ALA5133246 | nM | Rattus norvegicus | |||
| 2. |  ALA3211778 | SID57257030 | IC50 | = | 0.35 | uM | ALA4233686 | 6.46 | nM | Rattus norvegicus | ||
| 3. |  ALA271108 | 3 | Ki | = | 10.3 | nM | ALA4183542 | 7.99 | nM | Rattus norvegicus | ||
| 4. |  Tolterodine L-tartrate | Tolterodine | Ki | = | 3.6 | nM | ALA4183542 | 8.44 | nM | Rattus norvegicus | ||
| 5. |  ALA4745892 | Cyclostellettamine A | IC50 | = | 0.071 | mg/ml | ALA4676976 | ug.mL-1 | Rattus norvegicus | |||
| 6. |  ALA4788850 | Cyclostellettamine B | IC50 | = | 0.109 | mg/ml | ALA4676976 | ug.mL-1 | Rattus norvegicus | |||
| 7. |  ALA4743200 | Cyclostellettamine C | IC50 | = | 0.144 | mg/ml | ALA4676976 | ug.mL-1 | Rattus norvegicus | |||
| 8. |  ALA4749898 | Cyclostellettamine D | IC50 | = | 0.211 | mg/ml | ALA4676976 | ug.mL-1 | Rattus norvegicus | |||
| 9. |  ALA4750886 | Cyclostellettamine E | IC50 | = | 0.257 | mg/ml | ALA4676976 | ug.mL-1 | Rattus norvegicus | |||
| 10. |  ALA4797832 | Cyclostellettamine F | IC50 | = | 0.474 | mg/ml | ALA4676976 | ug.mL-1 | Rattus norvegicus | |||
| 11. |  ALA4795177 | 21g; VU6005806; AZN-00016130 | EC50 | > | 30 | uM | ALA4667452 | nM | Rattus norvegicus | |||
| 12. |  ALA4639776 | 9 | Activity | 0 | ALA4623764 | Dose-dependent effect | Rattus norvegicus | |||||
| 13. | ALA4639776 | 9 | Activity | = | 2.34 | g | ALA4623752 | g | Rattus norvegicus | |||
| 14. | ALA4639776 | 9 | Activity | = | 2.79 | g | ALA4623774 | g | Rattus norvegicus | |||
| 15. | ALA4639776 | 9 | Activity | = | 3.49 | g | ALA4623775 | g | Rattus norvegicus | |||
| 16. | ALA4639776 | 9 | FC | = | 158 | ALA4623758 | Rattus norvegicus | |||||
| 17. |  ALA4644670 | 8a; 4b | Ki | = | 0.47 | nM | ALA4605251 | 9.33 | nM | Rattus norvegicus | ||
| 18. |  4-Piperidyl n-(2-biphenyl)carbamate | 8a | Ki | = | 27 | nM | ALA4605251 | 7.57 | nM | Rattus norvegicus | ||
| 19. |  ML380 | 8n | EC50 | = | 3.1 | uM | ALA3370308 | 5.51 | nM | Rattus norvegicus | ||
| 20. |  ALA3298764 | 43a, ASP9133 | INH | 0 | ALA3369311 | Not Active | % | Rattus norvegicus |
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