# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY 678 | 17, BAY-678 | IC50 | > | 30 | uM | ALA5213837 | nM | Homo sapiens | |||
2. | ALA5198215 | Fig 2a, KLK5(1)-7 | Ki | = | 1.5 | nM | ALA5140186 | 8.82 | nM | Homo sapiens | ||
3. | ALA5185690 | Fig 2a, KLK5(1)-6 | Ki | = | 79 | nM | ALA5140186 | 7.10 | nM | Homo sapiens | ||
4. | ALA5176455 | Fig 2a, KLK5(1)-5 | Ki | = | 1.9 | nM | ALA5140186 | 8.72 | nM | Homo sapiens | ||
5. | ALA5174330 | Fig 2a, KLK5(1)-4 | Ki | = | 3.2 | nM | ALA5140186 | 8.49 | nM | Homo sapiens | ||
6. | ALA5205331 | Fig 2a, KLK5(1)-3 | Ki | = | 2.2 | nM | ALA5140186 | 8.66 | nM | Homo sapiens | ||
7. | ALA5194536 | Fig 2a, KLK5(1)-2 | Ki | = | 5.1 | nM | ALA5140186 | 8.29 | nM | Homo sapiens | ||
8. | ALA5175408 | Fig 2a, KLK5(1)-1 | Ki | = | 3.6 | nM | ALA5140186 | 8.44 | nM | Homo sapiens | ||
9. | ALA5199103 | Fig 2a, KLK5-7 | Ki | = | 1.4 | nM | ALA5140186 | 8.85 | nM | Homo sapiens | ||
10. | ALA5192991 | Fig 2a, KLK5-6 | Ki | = | 2.7 | nM | ALA5140186 | 8.57 | nM | Homo sapiens | ||
11. | ALA5175074 | Fig 2a, KLK5-5 | Ki | = | 29 | nM | ALA5140186 | 7.54 | nM | Homo sapiens | ||
12. | ALA5181364 | Fig 2a, KLK5-4 | Ki | = | 10.8 | nM | ALA5140186 | 7.97 | nM | Homo sapiens | ||
13. | ALA5203584 | Fig 2a, KLK5-3 | Ki | = | 29 | nM | ALA5140186 | 7.54 | nM | Homo sapiens | ||
14. | ALA5172150 | Fig 2a, KLK5-2 | Ki | = | 6.4 | nM | ALA5140186 | 8.19 | nM | Homo sapiens | ||
15. | ALA5194019 | Fig 2a, KLK5-1 | Ki | = | 5.8 | nM | ALA5140186 | 8.24 | nM | Homo sapiens | ||
16. | ALA5196523 | Fig 1b, R18C2 | Ki | = | 24 | nM | ALA5140186 | 7.62 | nM | Homo sapiens | ||
17. | ALA5172332 | Fig 1b, R13C2 | Ki | = | 28 | nM | ALA5140186 | 7.55 | nM | Homo sapiens | ||
18. | ALA5203034 | Fig 1b, R4C2 | Ki | = | 2.7 | nM | ALA5140186 | 8.57 | nM | Homo sapiens | ||
19. | ALA5209454 | Fig 1b, R20C1 | Ki | = | 6.1 | nM | ALA5140186 | 8.21 | nM | Homo sapiens | ||
20. | ALA5177587 | Fig 1b, R13C1 | Ki | = | 2 | nM | ALA5140186 | 8.70 | nM | Homo sapiens |