# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4214705 | 44; DKFZ-633 | Activity | 0 | ALA4201870 | Active | Homo sapiens | |||||
2. | ALA4214705 | 44; DKFZ-633 | Activity | 0 | ALA4201869 | Dose-dependent effect | Homo sapiens | |||||
3. | ALA4214705 | 44; DKFZ-633 | Activity | 0 | ALA4201868 | Active | Homo sapiens | |||||
4. | ALA4210314 | 42 | Activity | 0 | ALA4201868 | Active | Homo sapiens | |||||
5. | ALA4214705 | 44; DKFZ-633 | Activity | 0 | ALA4201867 | Active | Homo sapiens | |||||
6. | DKFZ‐251 | 11; DKFZ-251 | Activity | 0 | ALA4201862 | Dose-dependent effect | Homo sapiens | |||||
7. | DKFZ‐251 | 11; DKFZ-251 | Activity | 0 | ALA4201823 | Dose-dependent effect | Homo sapiens | |||||
8. | DKFZ‐251 | 11; DKFZ-251 | Activity | 0 | ALA4201860 | Active | Homo sapiens | |||||
9. | DKFZ‐251 | 11; DKFZ-251 | Activity | 0 | ALA4201854 | Dose-dependent effect | Homo sapiens | |||||
10. | DKFZ‐251 | 11; DKFZ-251 | IC50 | = | 0.47 | uM | ALA4201843 | 6.33 | nM | Homo sapiens | ||
11. | ALA4206734 | 39 | IC50 | = | 0.023 | uM | ALA4201843 | 7.64 | nM | Homo sapiens | ||
12. | DKFZ‐251 | 11; DKFZ-251 | t1/2 | = | 6.43 | hr | ALA4201840 | hr | Homo sapiens | |||
13. | ALA4212099 | 27 | t1/2 | = | 19.1 | hr | ALA4201840 | hr | Homo sapiens | |||
14. | ALA4205435 | 14 | t1/2 | < | 10 | min | ALA4201840 | hr | Homo sapiens | |||
15. | ALA4212332 | 1 | INH | 0 | ALA4201839 | Not Active | % | Homo sapiens | ||||
16. | ALA4212332 | 1 | TDI | 0 | ALA4201838 | Not Active | Homo sapiens | |||||
17. | DKFZ‐251 | 11; DKFZ-251 | Ratio | = | 1883 | /M/s | ALA4201837 | /M/s | Homo sapiens | |||
18. | DKFZ‐251 | 11; DKFZ-251 | Activity | 0 | ALA4201836 | Active | Homo sapiens | |||||
19. | ALA4212332 | 1 | Activity | 0 | ALA4201835 | Not Active | Homo sapiens | |||||
20. | ALA4212332 | 1 | Activity | 0 | ALA4201834 | Active | Homo sapiens |