# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA331943 | 1b | IC50 | > | 30 | uM | ALA2051716 | nM | Homo sapiens | |||
2. | 5-[[(3S)-3-[benzyl-(7-methoxynaphthalen-2-yl)sulfonylamino]-2-oxopyrrolidin-1-yl]methyl]thiophene-2-carboximidamide | 5 | IC50 | = | 1.5 | uM | ALA2051716 | 5.82 | nM | Homo sapiens | ||
3. | ALA2047315 | 4 | IC50 | = | 8.2 | uM | ALA2051716 | 5.09 | nM | Homo sapiens | ||
4. | ALA2047314 | 3 | IC50 | = | 2.9 | uM | ALA2051716 | 5.54 | nM | Homo sapiens | ||
5. | ALA435585 | 41 | IC50 | = | 7.75 | uM | ALA2051716 | 5.11 | nM | Homo sapiens | ||
6. | ALA331939 | 42 | IC50 | > | 30 | uM | ALA2051716 | nM | Homo sapiens | |||
7. | ALA4863579 | 46 | INH | = | 8.86 | % | ALA4831724 | % | Homo sapiens | |||
8. | ALA4846167 | 43 | INH | = | 19.81 | % | ALA4831724 | % | Homo sapiens | |||
9. | ALA4853958 | 38 | INH | = | 47 | % | ALA4831724 | % | Homo sapiens | |||
10. | ALA4848741 | 36 | INH | = | 21.83 | % | ALA4831724 | % | Homo sapiens | |||
11. | ALA4853857 | 35 | INH | = | 29.98 | % | ALA4831724 | % | Homo sapiens | |||
12. | ALA4865287 | 34 | INH | = | 7.27 | % | ALA4831724 | % | Homo sapiens | |||
13. | ALA4864566 | 33 | INH | = | 26.47 | % | ALA4831724 | % | Homo sapiens | |||
14. | ALA4846525 | 31 | INH | = | 20 | % | ALA4831724 | % | Homo sapiens | |||
15. | ALA4856926 | 30 | INH | = | 14.83 | % | ALA4831724 | % | Homo sapiens | |||
16. | ALA4862261 | 47 | Ki | = | 1 | uM | ALA4831723 | 6.00 | nM | Homo sapiens | ||
17. | ALA4852575 | 40 | Ki | = | 2.4 | uM | ALA4831723 | 5.62 | nM | Homo sapiens | ||
18. | ALA4863108 | 37 | Ki | = | 1.5 | uM | ALA4831723 | 5.82 | nM | Homo sapiens | ||
19. | ALA4847066 | 32 | Ki | = | 2 | uM | ALA4831723 | 5.70 | nM | Homo sapiens | ||
20. | ALA4853943 | 28 | Ki | = | 4.3 | uM | ALA4831723 | 5.37 | nM | Homo sapiens |