# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4748253 | 9 | INH | = | 99 | % | ALA4667691 | % | Homo sapiens | |||
2. | ALA4784899 | 51 | INH | = | -23.3 | % | ALA4667691 | % | Homo sapiens | |||
3. | ALA4789469 | 26 | INH | = | -28.8 | % | ALA4667691 | % | Homo sapiens | |||
4. | ALA3917415 | BDBM210853 | IC50 | = | 1043 | nM | ALA4049090 | 5.98 | nM | Homo sapiens | ||
5. | ALA4060249 | LSPN427, diastereomeric mixture 52:48 | INH | = | 3.9 | % | ALA4044518 | % | Homo sapiens | |||
6. | ALA4088774 | LSPN426, diastereomeric mixture 60:40 | INH | = | 21.3 | % | ALA4044518 | % | Homo sapiens | |||
7. | ALA4067529 | LSPN425, diastereomeric mixture 69:31 | INH | = | 0 | % | ALA4044518 | % | Homo sapiens | |||
8. | ALA4092481 | LSPN424, diastereomeric mixture 66:34 | INH | = | 0 | % | ALA4044518 | % | Homo sapiens | |||
9. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | INH | = | 30.8 | % | ALA4044518 | % | Homo sapiens | |||
10. | ALA4096825 | LSPN422, diastereomeric mixture 66:34 | INH | = | 43.5 | % | ALA4044518 | % | Homo sapiens | |||
11. | ALA4462944 | 43 | IC50 | = | 0.7 | uM | ALA4376337 | 6.16 | nM | Homo sapiens | ||
12. | ALA4438688 | 44 | IC50 | = | 0.42 | uM | ALA4376337 | 6.38 | nM | Homo sapiens | ||
13. | ALA4576261 | 45 | IC50 | = | 1.4 | uM | ALA4376337 | 5.85 | nM | Homo sapiens | ||
14. | ALA4566164 | 46 | INH | = | -16.1 | % | ALA4341510 | % | Homo sapiens | |||
15. | ALA4472283 | 44 | INH | = | 29.8 | % | ALA4341510 | % | Homo sapiens | |||
16. | ALA4459895 | 22 | INH | = | -28.7 | % | ALA4341510 | % | Homo sapiens | |||
17. | ALA4566164 | 46 | INH | = | 32.1 | % | ALA4341501 | % | Homo sapiens | |||
18. | ALA4472283 | 44 | INH | = | 58.4 | % | ALA4341501 | % | Homo sapiens | |||
19. | ALA4459895 | 22 | INH | = | 56.9 | % | ALA4341501 | % | Homo sapiens | |||
20. | ALA4566164 | 46 | INH | = | 86.3 | % | ALA4341492 | % | Homo sapiens |