# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4540759 | EUB0000545 | IC50 | > | 10 | uM | ALA4882308 | Not Active | nM | Homo sapiens | ||
2. | ALA2170610 | 60 | IC50 | > | 16 | uM | ALA4882308 | Not Active | nM | Homo sapiens | ||
3. | ALA3900457 | S-2120 | IC50 | = | 1.32 | uM | ALA3882221 | 5.88 | nM | Homo sapiens | ||
4. | ALA3897683 | S-3226 | IC50 | = | 0.02 | uM | ALA3882221 | 7.70 | nM | Homo sapiens | ||
5. | ALA3974005 | T-162559 (R) | IC50 | > | 30 | uM | ALA3882221 | nM | Homo sapiens | |||
6. | ALA3900790 | T-162559 (S) | IC50 | = | 11 | uM | ALA3882221 | 4.96 | nM | Homo sapiens | ||
7. | ALA51879 | 1a | IC50 | > | 30 | uM | ALA3882221 | nM | Homo sapiens | |||
8. | N-Carbamimidoyl-2-methyl-5-(methylsulfonyl)-4-(1H-pyrrol-1-yl)benzamide | 246 | IC50 | = | 100 | uM | ALA3882221 | 4.00 | nM | Homo sapiens | ||
9. | Cariporide | 267 | IC50 | >= | 1 | uM | ALA3882221 | nM | Homo sapiens | |||
10. | ALA3975004 | 005 | pIC50 | 0 | ALA3881404 | Not Determined | Homo sapiens | |||||
11. | ALA3911510 | 004 | pIC50 | = | 5.6 | ALA3881404 | 5.60 | nM | Homo sapiens | |||
12. | ALA3901000 | 003 | pIC50 | = | 8.1 | ALA3881404 | 8.10 | nM | Homo sapiens | |||
13. | Tenapanor hydrochloride | TENAPANOR HYDROCHLORIDE | pIC50 | = | 8.2 | ALA3881404 | 8.20 | nM | Homo sapiens | |||
14. | tenapanor | 180 | pIC50 | = | 8.3 | ALA3881394 | 8.30 | nM | Homo sapiens | |||
15. | ALA3961536 | 179 | pIC50 | = | 7.77 | ALA3881394 | 7.77 | nM | Homo sapiens | |||
16. | ALA3958849 | 178 | pIC50 | = | 7.33 | ALA3881394 | 7.33 | nM | Homo sapiens | |||
17. | ALA3902600 | 177 | pIC50 | = | 7.8 | ALA3881394 | 7.80 | nM | Homo sapiens | |||
18. | ALA3960033 | 176 | pIC50 | = | 7.4 | ALA3881394 | 7.40 | nM | Homo sapiens | |||
19. | ALA3945874 | 175 | pIC50 | = | 7.4 | ALA3881394 | 7.40 | nM | Homo sapiens | |||
20. | ALA3937928 | 174 | pIC50 | = | 8.53 | ALA3881394 | 8.53 | nM | Homo sapiens |