# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | N-Carbamimidoyl-2-methyl-5-(methylsulfonyl)-4-(1H-pyrrol-1-yl)benzamide | 246 | IC50 | > | 30 | uM | ALA4257134 | nM | Homo sapiens | |||
2. | Cariporide | 267 | IC50 | > | 30 | uM | ALA4257134 | nM | Homo sapiens | |||
3. | ALA51879 | 1a | IC50 | = | 3.36 | uM | ALA4257134 | 5.47 | nM | Homo sapiens | ||
4. | ALA466311 | 5l | IC50 | = | 0.37 | uM | ALA4257134 | 6.43 | nM | Homo sapiens | ||
5. | EIPA | EIPA | IC50 | = | 0.42 | uM | ALA4257134 | 6.38 | nM | Homo sapiens | ||
6. | Amiloride | 1 | IC50 | = | 21 | uM | ALA4257134 | 4.68 | nM | Homo sapiens | ||
7. | ALA51879 | 1a | IC50 | = | 3.36 | uM | ALA3882220 | 5.47 | nM | Homo sapiens | ||
8. | N-Carbamimidoyl-2-methyl-5-(methylsulfonyl)-4-(1H-pyrrol-1-yl)benzamide | 246 | IC50 | > | 30 | uM | ALA3882220 | nM | Homo sapiens | |||
9. | Cariporide | 267 | IC50 | > | 30 | uM | ALA3882220 | nM | Homo sapiens | |||
10. | 5-(N,N-Hexamethylene)amiloride | 5m | Ki | = | 0.37 | uM | ALA3882220 | 6.43 | nM | Homo sapiens | ||
11. | EIPA | EIPA | Ki | = | 0.42 | uM | ALA3882220 | 6.38 | nM | Homo sapiens | ||
12. | Amiloride | 1 | Ki | = | 21 | uM | ALA3882220 | 4.68 | nM | Homo sapiens | ||
13. | ALA51879 | 1a | IC50 | = | 3.36 | uM | ALA3881449 | 5.47 | nM | Homo sapiens | ||
14. | N-Carbamimidoyl-2-methyl-5-(methylsulfonyl)-4-(1H-pyrrol-1-yl)benzamide | 246 | IC50 | > | 30 | uM | ALA3881449 | nM | Homo sapiens | |||
15. | 5-(N,N-Hexamethylene)amiloride | 5m | Ki | = | 0.37 | uM | ALA3881449 | 6.43 | nM | Homo sapiens | ||
16. | Cariporide | 267 | IC50 | > | 30 | uM | ALA3881449 | nM | Homo sapiens | |||
17. | Amiloride | 1 | Ki | = | 21 | uM | ALA3881449 | 4.68 | nM | Homo sapiens | ||
18. | EIPA | EIPA | Ki | = | 0.42 | uM | ALA3881449 | 6.38 | nM | Homo sapiens | ||
19. | ALA3892788 | 13d.HCl | IC50 | = | 0.291 | uM | ALA3861050 | 6.54 | nM | Homo sapiens | ||
20. | ALA51879 | 1a | IC50 | = | 3.36 | uM | ALA748619 | 5.47 | nM | Homo sapiens |