# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GZD824 | 10a, GZD824 | IC50 | = | 2.08 | nM | ALA5241432 | 8.68 | nM | Homo sapiens | ||
2. | ALA4278642 | 25e; SOMCL-085 | IC50 | = | 22.6 | nM | ALA5241387 | 7.65 | nM | Homo sapiens | ||
3. | AZD3229 | 44; AZD3229 | IC50 | = | 1 | nM | ALA5238318 | 9.00 | nM | Homo sapiens | ||
4. | Ripretinib (DCC-2618) | 4; DCC-2618 | IC50 | = | 36 | uM | ALA5238317 | 4.44 | nM | Homo sapiens | ||
5. | ALA5274267 | 8u | IC50 | > | 10 | uM | ALA5226043 | nM | Homo sapiens | |||
6. | CLK-IN-T3 | EUB0000321 | IC50 | = | 2.52 | uM | ALA5213256 | 5.60 | nM | Homo sapiens | ||
7. | CLK-IN-T3 | EUB0000321 | % of control | = | 29 | % | ALA5213255 | % | Homo sapiens | |||
8. | BMS-777607 | 10, BMS-777607 | % of control | = | 0.2 | % | ALA5212877 | % | Homo sapiens | |||
9. | GSK461364 | GSK-461364A | % of inhibition | = | 96 | % | ALA5214851 | % | Homo sapiens | |||
10. | BIX 02565 | 24, BIX 02565, eutamer | IC50 | = | 956 | nM | ALA5213144 | 6.02 | nM | Homo sapiens | ||
11. | ALA5201881 | 30 | INH | < | 50 | % | ALA5167151 | % | Homo sapiens | |||
12. | ALA5193819 | 24 | INH | < | 50 | % | ALA5167151 | % | Homo sapiens | |||
13. | ALA5175977 | 28 | IC50 | > | 10 | uM | ALA5165271 | nM | Homo sapiens | |||
14. | PF-543 | PF-543 | IC50 | > | 10 | uM | ALA5165271 | nM | Homo sapiens | |||
15. | Afatinib | BIBW-2992 | IC50 | > | 10000 | nM | ALA5161047 | nM | Homo sapiens | |||
16. | ALA5208454 | C6 | IC50 | > | 10000 | nM | ALA5161047 | nM | Homo sapiens | |||
17. | ALA5182567 | C5 | IC50 | > | 10000 | nM | ALA5161047 | nM | Homo sapiens | |||
18. | ALA5184634 | 7m | Activity | 0 | ALA5160597 | Active | Homo sapiens | |||||
19. | ALA5177453 | 7b | IC50 | = | 102.4 | nM | ALA5160550 | 6.99 | nM | Homo sapiens | ||
20. | ALA5206811 | 7c | IC50 | = | 73.6 | nM | ALA5160550 | 7.13 | nM | Homo sapiens |