# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Entacapone | 1 (entacapone) | pIC50 | = | 8.52 | ALA4432181 | 8.52 | nM | Rattus norvegicus | |||
2. | Tolcapone | Tolcapone | pIC50 | = | 9.04 | ALA4432181 | 9.04 | nM | Rattus norvegicus | |||
3. | ALA4543735 | 25 | pIC50 | = | 8.43 | ALA4432181 | 8.43 | nM | Rattus norvegicus | |||
4. | ALA4444830 | 24 | pIC50 | = | 8.32 | ALA4432181 | 8.32 | nM | Rattus norvegicus | |||
5. | ALA481644 | III-26 | pIC50 | = | 8.31 | ALA4432181 | 8.31 | nM | Rattus norvegicus | |||
6. | ALA4447349 | 22 | pIC50 | = | 8.73 | ALA4432181 | 8.73 | nM | Rattus norvegicus | |||
7. | Caffeic acid | 28 | IC50 | = | 5861 | nM | ALA4432180 | 5.23 | nM | Rattus norvegicus | ||
8. | Caffeic acid phenethyl ester | CAPE | IC50 | 0 | ALA4432180 | Not Active | Rattus norvegicus | |||||
9. | ALA133714 | 13 | IC50 | 0 | ALA4432180 | Not Active | Rattus norvegicus | |||||
10. | ALA137555 | 7 | IC50 | = | 12.84 | nM | ALA4432180 | 7.89 | nM | Rattus norvegicus | ||
11. | Tyrphostin AG 1290 | 9 | IC50 | = | 55.35 | nM | ALA4432180 | 7.26 | nM | Rattus norvegicus | ||
12. | ALA4437043 | 19 | IC50 | = | 11.35 | nM | ALA4432180 | 7.95 | nM | Rattus norvegicus | ||
13. | ALA4463709 | 20 | IC50 | = | 12.82 | nM | ALA4432180 | 7.89 | nM | Rattus norvegicus | ||
14. | ALA4472878 | 21 | IC50 | = | 329.34 | nM | ALA4432180 | 6.48 | nM | Rattus norvegicus | ||
15. | ALA4447349 | 22 | IC50 | = | 52.47 | nM | ALA4432180 | 7.28 | nM | Rattus norvegicus | ||
16. | ALA481644 | III-26 | IC50 | = | 124.87 | nM | ALA4432180 | 6.90 | nM | Rattus norvegicus | ||
17. | ALA4444830 | 24 | IC50 | = | 137.6 | nM | ALA4432180 | 6.86 | nM | Rattus norvegicus | ||
18. | ALA4543735 | 25 | IC50 | = | 64.81 | nM | ALA4432180 | 7.19 | nM | Rattus norvegicus | ||
19. | ALA4448310 | 26 | IC50 | = | 29.86 | nM | ALA4432180 | 7.53 | nM | Rattus norvegicus | ||
20. | ALA4437795 | 27 | IC50 | = | 54.85 | nM | ALA4432180 | 7.26 | nM | Rattus norvegicus |