# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 50 | uM | ALA5252861 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 50 | uM | ALA5252861 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 50 | uM | ALA5252861 | nM | Homo sapiens | |||
4. | ALA4213175 | Fig S3, Cpd 6 | IC50 | > | 50 | uM | ALA5252861 | nM | Homo sapiens | |||
5. | ALA5270781 | 38 | IC50 | = | 0.36 | uM | ALA5252021 | 6.44 | nM | Homo sapiens | ||
6. | ALA5288241 | B2 | INH | = | 74 | % | ALA5238238 | % | Homo sapiens | |||
7. | Enzastaurin (LY317615) | 1e | Kd | = | 36 | nM | ALA5214809 | 7.44 | nM | Homo sapiens | ||
8. | NTQ1062 | 22b; NTQ1062 | INH | = | 90 | % | ALA5168708 | % | Homo sapiens | |||
9. | Tozasertib | VX-680 | INH | = | 5 | % | ALA5159034 | % | Homo sapiens | |||
10. | Sotrastaurin | 1 | INH | = | 99 | % | ALA5159034 | % | Homo sapiens | |||
11. | ALA494314 | 4g | IC50 | = | 2.8 | uM | ALA5159020 | 5.55 | nM | Homo sapiens | ||
12. | Sotrastaurin | 1 | IC50 | = | 0.22 | nM | ALA5159020 | 9.66 | nM | Homo sapiens | ||
13. | ALA5203363 | 2n | INH | = | 97 | % | ALA5158991 | % | Homo sapiens | |||
14. | ALA5196716 | 2m | INH | = | 60 | % | ALA5158991 | % | Homo sapiens | |||
15. | ALA5206391 | 2l | INH | = | 85 | % | ALA5158991 | % | Homo sapiens | |||
16. | ALA5170735 | 2k | INH | = | 7 | % | ALA5158991 | % | Homo sapiens | |||
17. | ALA5198734 | 2j | INH | = | 14 | % | ALA5158991 | % | Homo sapiens | |||
18. | ALA5185816 | 2i | INH | = | 83 | % | ALA5158991 | % | Homo sapiens | |||
19. | ALA5188904 | 2h | INH | = | 12 | % | ALA5158991 | % | Homo sapiens | |||
20. | ALA5189743 | 2g | INH | = | 25 | % | ALA5158991 | % | Homo sapiens |