# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | XL041 | BMS-852927 | PB | = | 97.3 | % | ALA3868535 | % | Homo sapiens | |||
2. | ALA3953927 | 13 | PB | = | 87.6 | % | ALA3868535 | % | Homo sapiens | |||
3. | ALA3944154 | 10 | PB | = | 86.6 | % | ALA3868535 | % | Homo sapiens | |||
4. | ALA3913162 | 8 | PB | = | 90.2 | % | ALA3868535 | % | Homo sapiens | |||
5. | ALA3890276 | 6 | PB | = | 99 | % | ALA3868535 | % | Homo sapiens | |||
6. | BMS-779788 | 18 | PB | = | 99.9 | % | ALA3868535 | % | Homo sapiens | |||
7. | Primaquine bisphosphate | Primaquine diphosphate | Ka | = | 8 | 10^5/M | ALA936356 | 10^5/M | Homo sapiens | |||
8. | ALA3216010 | amodiaquine diHCl | Ka | = | 5.8 | 10^4/M | ALA936356 | 10^4/M | Homo sapiens | |||
9. | ALA523 | 3 | Activity | = | 9 | uM | ALA905138 | uM | Homo sapiens | |||
10. | ALA387720 | 3 | Activity | = | 14 | uM | ALA905138 | uM | Homo sapiens | |||
11. | ALA229118 | 4 | Activity | = | 13 | uM | ALA905138 | uM | Homo sapiens | |||
12. | Diazepam | Diazepam | Activity | = | 10 | uM | ALA905138 | uM | Homo sapiens | |||
13. | Cetirizine | 66 ((R)cetirizine) | Ka | = | 5.12 | M/M | ALA623839 | M/M | Homo sapiens | |||
14. | Cetirizine | 66 ((R)cetirizine) | n | = | 1.74 | ALA623840 | Homo sapiens | |||||
15. | ALA288292 | 15 | Inhibition | = | 42 | % | ALA644688 | % | Homo sapiens | |||
16. | ALA288811 | 13 | IC50 | = | 5 | mM | ALA644687 | nM | Homo sapiens | |||
17. | ALA375586 | sLex | IC50 | = | 8 | mM | ALA644687 | nM | Homo sapiens | |||
18. | ALA287905 | 14 | Inhibition | = | 45 | % | ALA644688 | % | Homo sapiens | |||
19. | ALA432294 | 16 | Inhibition | = | 43 | % | ALA644688 | % | Homo sapiens |