# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2012574 | 42, LDN-211898 | INH | = | 34 | % | ALA2015474 | % | Homo sapiens | |||
2. | BAY-091 | EUB0001564 | % inhibition | 9.88 | % | ALA4887994 | Not Active | % | Homo sapiens | |||
3. | ALA4580220 | EUB0000311 | % residual kinase activity | 101 | % | ALA4884427 | Not Active | % | Homo sapiens | |||
4. | BAY-885 | BAY-885; 41 | % residual kinase activity | 104 | % | ALA4881175 | Not Active | % | Homo sapiens | |||
5. | ALA3354665 | 11a | IC50 | = | 1.743 | uM | ALA3378296 | 5.76 | nM | Homo sapiens | ||
6. | ALA4860270 | 17 | INH | = | 3.1 | % | ALA4824988 | % | Homo sapiens | |||
7. | ALA4876923 | 16 | INH | = | 34 | % | ALA4824988 | % | Homo sapiens | |||
8. | ALA4870610 | 15 | INH | = | 45 | % | ALA4824988 | % | Homo sapiens | |||
9. | ALA4848708 | 14 | INH | = | 17 | % | ALA4824988 | % | Homo sapiens | |||
10. | ALA4847931 | 11 | INH | = | 8.5 | % | ALA4824988 | % | Homo sapiens | |||
11. | ALA4877843 | 8 | INH | = | 20 | % | ALA4824988 | % | Homo sapiens | |||
12. | ALA4847005 | 6 | INH | = | 40 | % | ALA4824988 | % | Homo sapiens | |||
13. | ALA4857154 | 4 | INH | = | 50 | % | ALA4824988 | % | Homo sapiens | |||
14. | 3,3-Dimethylindolin-2-one | 2 | INH | = | 8 | % | ALA4824988 | % | Homo sapiens | |||
15. | ALA4860270 | 17 | IC50 | > | 30 | uM | ALA4824986 | nM | Homo sapiens | |||
16. | ALA4876923 | 16 | IC50 | > | 100 | uM | ALA4824986 | nM | Homo sapiens | |||
17. | ALA4870610 | 15 | IC50 | > | 30 | uM | ALA4824986 | nM | Homo sapiens | |||
18. | ALA4848708 | 14 | IC50 | > | 30 | uM | ALA4824986 | nM | Homo sapiens | |||
19. | ALA4847931 | 11 | IC50 | > | 30 | uM | ALA4824986 | nM | Homo sapiens | |||
20. | ALA4877843 | 8 | IC50 | > | 300 | uM | ALA4824986 | nM | Homo sapiens |