# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5279874 | 28 | IC50 | = | 40 | uM | ALA5242032 | 4.40 | nM | Homo sapiens | ||
2. | ALA5273669 | 51 | IC50 | = | 0.9 | nM | ALA5232760 | 9.05 | nM | Homo sapiens | ||
3. | ALA5290077 | 50 | IC50 | = | 4.6 | nM | ALA5232760 | 8.34 | nM | Homo sapiens | ||
4. | ALA5280395 | 49 | IC50 | = | 1.9 | nM | ALA5232760 | 8.72 | nM | Homo sapiens | ||
5. | ALA5281180 | 48 | IC50 | = | 12 | nM | ALA5232760 | 7.92 | nM | Homo sapiens | ||
6. | ALA5282677 | 47 | IC50 | = | 0.9 | nM | ALA5232760 | 9.05 | nM | Homo sapiens | ||
7. | ALA5283969 | 46 | IC50 | > | 50000 | nM | ALA5232760 | nM | Homo sapiens | |||
8. | Forodesine | 1 | IC50 | = | 0.06 | nM | ALA5232760 | 10.22 | nM | Homo sapiens | ||
9. | ALA475750 | 4, DADMe-ImmG | Ki | = | 7 | pM | ALA4377146 | nM | Homo sapiens | |||
10. | Ulodesine | DADMe-ImmH | Ki | = | 16 | pM | ALA4377146 | 10.80 | nM | Homo sapiens | ||
11. | ALA475750 | 4, DADMe-ImmG | Ki | = | 0.16 | nM | ALA4377145 | 9.80 | nM | Homo sapiens | ||
12. | Ulodesine | DADMe-ImmH | Ki | = | 1.1 | nM | ALA4377145 | 8.96 | nM | Homo sapiens | ||
13. | Inosine | Inosine | Kcat | = | 56 | /s | ALA4377120 | /s | Homo sapiens | |||
14. | ALA473929 | 2, MeS-ImmH | Ki | = | 303 | nM | ALA4377143 | 6.52 | nM | Homo sapiens | ||
15. | ALA474121 | 5, L-ImmH | Ki | = | 9 | nM | ALA4377141 | 8.05 | nM | Homo sapiens | ||
16. | ALA454743 | 6, L-DADMe-ImmH | Ki | = | 80 | nM | ALA4377141 | 7.10 | nM | Homo sapiens | ||
17. | ALA473922 | 2 | Ki | = | 29 | nM | ALA4377141 | nM | Homo sapiens | |||
18. | Forodesine | 1 | Ki | = | 72 | nM | ALA4377141 | nM | Homo sapiens | |||
19. | ALA474121 | 5, L-ImmH | Ki | = | 32 | nM | ALA4377140 | 7.50 | nM | Homo sapiens | ||
20. | ALA454743 | 6, L-DADMe-ImmH | Ki | = | 1700 | nM | ALA4377140 | 5.77 | nM | Homo sapiens |