# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3785951 | 33 | IC50 | > | 10 | uM | ALA3790310 | nM | Homo sapiens | |||
2. | ALA3786167 | 28 | IC50 | > | 10 | uM | ALA3790310 | nM | Homo sapiens | |||
3. | ALA3785500 | 3 | IC50 | > | 10 | uM | ALA3790310 | nM | Homo sapiens | |||
4. | ALA3787112 | 2 | IC50 | = | 1.5 | uM | ALA3790310 | 5.82 | nM | Homo sapiens | ||
5. | ALA3787614 | 17 | IC50 | > | 10 | uM | ALA3790310 | nM | Homo sapiens | |||
6. | ALA1614712 | 1; NVP-AEW541 | IC50 | > | 10 | uM | ALA3790310 | nM | Homo sapiens | |||
7. | ALA3780032 | 5; IACS-4759 | INH | 0 | ALA3782403 | Not Active | % | Homo sapiens | ||||
8. | ALA3782012 | 1 | IC50 | = | 60 | nM | ALA3784141 | 7.22 | nM | Homo sapiens | ||
9. | ALA3781427 | 2 | IC50 | = | 9 | nM | ALA3784141 | 8.05 | nM | Homo sapiens | ||
10. | ALA3780091 | 10 | IC50 | = | 1.5 | nM | ALA3784141 | 8.82 | nM | Homo sapiens | ||
11. | ALA3780467 | 21 | IC50 | = | 7 | nM | ALA3784141 | 8.15 | nM | Homo sapiens | ||
12. | Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 0.72 | nM | ALA3784141 | 9.14 | nM | Homo sapiens | ||
13. | racemic-tofacitinib | CP-690550 | IC50 | = | 12.8 | nM | ALA3784141 | 7.89 | nM | Homo sapiens | ||
14. | ALA3771285 | 12 | Activity | = | 94 | % | ALA3772131 | % | Homo sapiens | |||
15. | ALA3764637 | 9 | IC50 | = | 310 | nM | ALA3766659 | 6.51 | nM | Homo sapiens | ||
16. | ALA3764167 | 10 | IC50 | = | 650 | nM | ALA3766659 | 6.19 | nM | Homo sapiens | ||
17. | ALA3763697 | 11 | IC50 | = | 1100 | nM | ALA3766659 | 5.96 | nM | Homo sapiens | ||
18. | ALA3763184 | 12 | IC50 | = | 6900 | nM | ALA3766659 | 5.16 | nM | Homo sapiens | ||
19. | ALA3763252 | 13 | IC50 | = | 54 | nM | ALA3766659 | 7.27 | nM | Homo sapiens | ||
20. | ALA3763991 | 14 | IC50 | = | 48 | nM | ALA3766659 | 7.32 | nM | Homo sapiens |