# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5274306 | 15 | INH | < | 50 | % | ALA5228839 | % | Homo sapiens | |||
2. | ALA5274312 | 26; MRS4853 | Ki | = | 3.5 | uM | ALA5224977 | 5.46 | nM | Homo sapiens | ||
3. | ALA4576555 | EUB0000705 | Ki | = | 1901 | nM | ALA5213384 | 5.72 | nM | Homo sapiens | ||
4. | CLK-IN-T3 | EUB0000321 | Ki | = | 2154.79 | nM | ALA5213241 | 5.67 | nM | Homo sapiens | ||
5. | ALA3337895 | 26f | Ki | = | 19 | nM | ALA5213655 | 7.72 | nM | Homo sapiens | ||
6. | ALA3337894 | 26c | Ki | = | 98 | nM | ALA5213675 | 7.01 | nM | Homo sapiens | ||
7. | NVS-PAK1-1 | 3 | IC50 | = | 13 | uM | ALA5213589 | 4.89 | nM | Homo sapiens | ||
8. | ALA4561806 | EUB0001135 | % of inhibition | = | 49.9 | % | ALA5213906 | % | Homo sapiens | |||
9. | ALA4552180 | EUB0000251 | % of inhibition | = | 46 | % | ALA5214492 | % | Homo sapiens | |||
10. | BAY 293 Negative Control | EUB0000743 | Ki | = | 1365.75 | nM | ALA5213957 | 5.87 | nM | Homo sapiens | ||
11. | ALA4761843 | EUB0000348aPTSA | Ki | > | 10 | uM | ALA5214401 | nM | Homo sapiens | |||
12. | ALA4761843 | EUB0000348aPTSA | % of inhibition | = | 54 | % | ALA5214400 | % | Homo sapiens | |||
13. | ALA4513786 | ABT-546 | Ki | > | 10 | uM | ALA5213812 | nM | Homo sapiens | |||
14. | A192621 | 38 | % of inhibition | = | 35.99 | % | ALA5214407 | % | Homo sapiens | |||
15. | A-1155463 | 17, A-1155463 | % of inhibition | = | 69.2 | % | ALA5213785 | % | Homo sapiens | |||
16. | A-1155463 | 17, A-1155463 | % of inhibition | = | 69.2 | % | ALA5213784 | % | Homo sapiens | |||
17. | doxepin | SID11111071 | pKi | = | 9.75 | ALA5169022 | 9.75 | nM | Homo sapiens | |||
18. | ALA5175488 | 1 | pKd | = | 8.1 | ALA5169021 | 8.10 | nM | Homo sapiens | |||
19. | ALA5192377 | 39f | Activity | 0 | ALA5169016 | Active | Homo sapiens | |||||
20. | ALA5189492 | 39d | Activity | 0 | ALA5169016 | Active | Homo sapiens |