# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | conivaptan | Conivaptan | Ki | > | 10000 | nM | ALA4201577 | nM | Rattus norvegicus | |||
2. | ALA1253499 | 13, SSR-126768A | Ki | = | 46 | nM | ALA1253136 | 7.34 | nM | Rattus norvegicus | ||
3. | ALA1223814 | 24 | IC50 | = | 0.21 | uM | ALA1225851 | 6.68 | nM | Rattus norvegicus | ||
4. | SSR 149415 | 1, SSR-149415 | Ki | = | 1 | nM | ALA1686968 | 9.00 | nM | Rattus norvegicus | ||
5. | ALA1684574 | 12j | IC50 | = | 4 | nM | ALA1686968 | 8.40 | nM | Rattus norvegicus | ||
6. | ALA1684573 | 12i | IC50 | = | 2 | nM | ALA1686968 | 8.70 | nM | Rattus norvegicus | ||
7. | ALA221485 | 1 | Activity | = | 73 | % | ALA907389 | Agonist | % | Rattus norvegicus | ||
8. | ALA412742 | 3 | Activity | = | 97 | % | ALA907389 | Agonist | % | Rattus norvegicus | ||
9. | ALA265859 | B | Activity | = | 128 | % | ALA907389 | Agonist | % | Rattus norvegicus | ||
10. | d[Leu4,Lys8]-VP | 5 | Activity | = | 124 | % | ALA907389 | Agonist | % | Rattus norvegicus | ||
11. | ALA373968 | 8 | Activity | = | 108 | % | ALA907389 | Agonist | % | Rattus norvegicus | ||
12. | d[Cha4]-AVP | d[Cha4]AVP | Activity | = | 110 | % | ALA907389 | Agonist | % | Rattus norvegicus | ||
13. | d[Cha4]-AVP | d[Cha4]AVP | Kact | = | 0.6 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
14. | ALA221485 | 1 | Kact | = | 2.7 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
15. | ALA412742 | 3 | Kact | = | 1.4 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
16. | ALA265859 | B | Kact | = | 0.4 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
17. | d[Leu4,Lys8]-VP | 5 | Kact | = | 1.5 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
18. | ALA373968 | 8 | Kact | = | 1.6 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
19. | Argipressin | AVP | Kact | = | 2.3 | nM | ALA907388 | Agonist | nM | Rattus norvegicus | ||
20. | d[Cha4]-AVP | d[Cha4]AVP | Ki | = | 1.4 | nM | ALA907379 | 8.85 | Antagonist | nM | Rattus norvegicus |