# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3527569 | M25 | Drug metabolism | 0 | ALA3540072 | metabolite_detected | Homo sapiens | |||||
2. | Brivanib (BMS-540215) | 12 | Drug metabolism | 0 | ALA3539756 | metabolite_detected | Homo sapiens | |||||
3. | ALA1402 | 3 | Km(app) | = | 6.4 | uM | ALA3540602 | nM | Homo sapiens | |||
4. | ALA1402 | 3 | Vmax | = | 5.5 | nmol/min | ALA3540605 | nmol/min | Homo sapiens | |||
5. | β-Estradiol | Table II | Km | = | 4 | nM | ALA3537877 | nM | Homo sapiens | |||
6. | ALA4753179 | 2 | IC50 | = | 19.8 | uM | ALA4701345 | 4.70 | nM | Homo sapiens | ||
7. | ALA4551402 | 25 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
8. | ALA503833 | 6b | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
9. | ALA4564405 | 23 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
10. | ALA4517100 | 22 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
11. | ALA4560974 | 21 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
12. | ALA4576000 | 20 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
13. | ALA490084 | 3b | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
14. | ALA4525617 | 18 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
15. | ALA4557856 | 17 | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
16. | 2-(4-Aminophenyl)benzo[d]thiazol-6-ol | 6-Substituted BTA analogue | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
17. | ALA91449 | 6-Substituted BTA analogue | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
18. | 2-(4-(Methylamino)phenyl)benzo[d]thiazol-6-ol | 6-Substituted BTA analogue | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
19. | ALA47361 | 3g | Vmax/Km | 0 | ALA4482700 | Bld | Homo sapiens | |||||
20. | 2-Methyl-5-benzothiazolol | 12 | Vmax/Km | = | 0.01 | ALA4482700 | Homo sapiens |