# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2419769 | (S)-6 | pA2 | = | 9.01 | ALA2422340 | 9.01 | nM | Rattus norvegicus | |||
2. | ALA2419771 | (S)-8 | pA2 | = | 9.58 | ALA2422340 | 9.58 | nM | Rattus norvegicus | |||
3. | ALA2419765 | (S)-7 | pA2 | = | 8.52 | ALA2422340 | 8.52 | nM | Rattus norvegicus | |||
4. | ALA3216590 | (S)-9 | pA2 | = | 8.62 | ALA2422340 | 8.62 | nM | Rattus norvegicus | |||
5. | BMY 7378 dihydrochloride | BMY-7378 | pA2 | = | 8.34 | ALA2422340 | 8.34 | nM | Rattus norvegicus | |||
6. | ALA2407174 | 7 | INH | = | 31 | % | ALA2411859 | % | Rattus norvegicus | |||
7. | ALA1259203 | 7 | INH | > | 50 | % | ALA2327479 | % | Rattus norvegicus | |||
8. | Sertindole | 14c | Ki | = | 0.66 | nM | ALA2327486 | 9.18 | nM | Rattus norvegicus | ||
9. | ALA319352 | 12a | Ki | = | 2 | nM | ALA2327486 | 8.70 | nM | Rattus norvegicus | ||
10. | ALA328187 | 8a | Ki | = | 8.6 | nM | ALA2327486 | 8.07 | nM | Rattus norvegicus | ||
11. | ALA1259203 | 7 | Ki | = | 2.5 | nM | ALA2327486 | 8.60 | nM | Rattus norvegicus | ||
12. | ALA2326175 | 3l | Ki | = | 15 | nM | ALA2327486 | 7.82 | nM | Rattus norvegicus | ||
13. | ALA2261604 | (+)-1 | pA2 | = | 7.27 | ALA3058311 | 7.27 | nM | Rattus norvegicus | |||
14. | ALA2261605 | (+)-2 | pA2 | = | 7.23 | ALA3058311 | 7.23 | nM | Rattus norvegicus | |||
15. | ALA2261606 | (+)-3 | pA2 | = | 7.04 | ALA3058311 | 7.04 | nM | Rattus norvegicus | |||
16. | ALA2261607 | (+)-4 | pA2 | = | 7.05 | ALA3058311 | 7.05 | nM | Rattus norvegicus | |||
17. | ALA2261608 | (+)-5 | pA2 | = | 6.67 | ALA3058311 | 6.67 | nM | Rattus norvegicus | |||
18. | ALA2261604 | (+)-1 | pA2 | = | 6.86 | ALA3056383 | 6.86 | nM | Rattus norvegicus | |||
19. | ALA61006 | 1 | pKi | = | 5.07 | ALA3056710 | 5.07 | nM | Rattus norvegicus | |||
20. | 2-Amino-1-(2,5-dimethoxyphenyl)ethanol | 5 | pKi | = | 5.78 | ALA3056710 | 5.78 | nM | Rattus norvegicus |