# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1182155 | (S)-1 | pKi | = | 8.24 | ALA5245781 | 8.24 | nM | Homo sapiens | |||
2. | ALA5274306 | 15 | INH | < | 50 | % | ALA5228823 | % | Homo sapiens | |||
3. | PFI-3 | 72; PFI-3 | IC50 | = | 3.6 | uM | ALA5214135 | 5.44 | nM | Homo sapiens | ||
4. | ALA4745071 | EUB0000337aCl | Ki | = | 3602 | nM | ALA5214342 | 5.44 | nM | Homo sapiens | ||
5. | ALA4752561 | EUB0000739a | Ki | > | 10000 | nM | ALA5213898 | nM | Homo sapiens | |||
6. | GSK343 | 6, GSK343 | IC50 | = | 10 | uM | ALA5214633 | 5.00 | nM | Homo sapiens | ||
7. | BIX 02565 | 24, BIX 02565, eutamer | IC50 | = | 52 | nM | ALA5213135 | 7.28 | nM | Homo sapiens | ||
8. | BAY 293 Negative Control | EUB0000743 | Ki | = | 95.26 | nM | ALA5213949 | 7.02 | nM | Homo sapiens | ||
9. | (S)-ZINC 3573 | EUB0000345 | Ki | = | 2294 | nM | ALA5214385 | 5.64 | nM | Homo sapiens | ||
10. | ALA4762646 | EUB0000341aCl | IC50 | = | 1.2 | uM | ALA5214367 | 5.92 | nM | Homo sapiens | ||
11. | ALA4753450 | EUB0000300bCl | Ki | > | 1.2 | uM | ALA5214433 | nM | Homo sapiens | |||
12. | ALA4594433 | ML-246 | Activity | < | 50 | % | ALA5168972 | % | Homo sapiens | |||
13. | RLX-33 | 33 | INH | < | 50 | % | ALA5167516 | % | Homo sapiens | |||
14. | ALA5182943 | 107 | INH | < | 50 | % | ALA5135874 | % | Homo sapiens | |||
15. | ALA5207529 | 106 | INH | < | 50 | % | ALA5135874 | % | Homo sapiens | |||
16. | ALA5204071 | 94 | INH | < | 50 | % | ALA5135874 | % | Homo sapiens | |||
17. | ALA5170784 | 93 | INH | < | 50 | % | ALA5135874 | % | Homo sapiens | |||
18. | ALA5201983 | 12 | Ki | = | 11 | nM | ALA5117898 | 7.96 | nM | Homo sapiens | ||
19. | ALA5191141 | 10; Lu AF35700 | Ki | = | 2.9 | nM | ALA5117898 | 8.54 | nM | Homo sapiens | ||
20. | ALA4446822 | 14 | Activity | = | 22.28 | % | ALA4416566 | % | Homo sapiens |