| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4442951 | DHD3; D2 | Activity | = | 84 | % | ALA4378688 | % | Homo sapiens | |||
| 2. | ALA4442951 | DHD3; D2 | CL | < | 2.9 | uL/min/pmol | ALA4378676 | uL/min/pmol | Homo sapiens | |||
| 3. |  ALA4550375 | DHD1; D1 | CL | < | 2.9 | uL/min/pmol | ALA4378676 | uL/min/pmol | Homo sapiens | |||
| 4. |  PDK4-IN-1 hydrochloride | 8c | IC50 | > | 50 | uM | ALA4333065 | nM | Homo sapiens | |||
| 5. |  PT-2385 | (S)-10i | Drug metabolism | 0 | ALA4312545 | Metabolite_Notdetected | Homo sapiens | |||||
| 6. |  PF-05221304 | 38 | IC50 | > | 20 | uM | ALA4669914 | nM | Homo sapiens | |||
| 7. |  ALA3398252 | 2 | Drug metabolism | 0 | ALA3398973 | metabolite_notdetected | Homo sapiens | |||||
| 8. |  Raltegravir (MK-0518) | 1, raltegravir | Drug metabolism | 0 | ALA3398973 | metabolite_detected | Homo sapiens | |||||
| 9. | ALA3398252 | 2 | Activity | 0 | ALA3398978 | Not Active | Homo sapiens | |||||
| 10. | ALA3398252 | 2 | IC50 | 0 | ALA3399064 | Not Active | Homo sapiens | |||||
| 11. | ALA3398252 | 2 | Activity | 0 | ALA3399068 | Active | Homo sapiens | |||||
| 12. |  1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3531832 | metabolite_not_detected | Homo sapiens | |||||
| 13. |  ALA3527359 | YM150 monomaleate | Drug metabolism | < | 0.01 | nmol/min | ALA3534354 | nmol/min | Homo sapiens | |||
| 14. |  Haloperidol | Haloperidol | Drug metabolism | = | 120 | % | ALA3534013 | % | Homo sapiens | |||
| 15. | Haloperidol | Haloperidol | Drug metabolism | = | 99 | % | ALA3529643 | % | Homo sapiens | |||
| 16. | Haloperidol | Haloperidol | Drug metabolism | = | 4 | % | ALA3537959 | % | Homo sapiens | |||
| 17. |  ALA1710 | TFP HCl | Drug metabolism | = | 0.26 | nmol/min/mg | ALA3537956 | nmol/min/mg | Homo sapiens | |||
| 18. |  Dolutegravir (GSK1349572) | DOLUTEGRAVIR | Drug metabolism | 0 | ALA3541848 | metabolite_not_detected | Homo sapiens | |||||
| 19. | Haloperidol | Haloperidol | CL | = | 9 | uL/min/g | ALA3540230 | mL.min-1.g-1 | Homo sapiens | |||
| 20. | Haloperidol | Haloperidol | Vmax | = | 0.6 | nmol/min | ALA3540229 | nmol/min | Homo sapiens |
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