| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Tamoxifen | Tamoxifen | Vmax | = | 402 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 2. |  ALA715 | Olanzapine | Vmax | = | 2370 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 3. |  ketotifen | ketotifen | Vmax | = | 140 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 4. | ketotifen | ketotifen | Vmax | = | 130 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 5. |  Imipramine | Imipramine | Vmax | = | 180 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 6. |  α-Hydroxy Tamoxifen | cis-Hydroxy-tamoxifen | Vmax | = | 547 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 7. | α-Hydroxy Tamoxifen | cis-Hydroxy-tamoxifen | Vmax | = | 315 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 8. |  ALA837 | 44 | Vmax | = | 132 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 9. |  cyproheptadine | 7 | Vmax | = | 49 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 10. |  ALA1908108 | C-posaconazole | Vmax | = | 17 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 11. |  Amitriptyline | Amitriptyline | Vmax | = | 96 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 12. | Amitriptyline | Amitriptyline | Vmax | = | 340 | pmol/min/mg protein | ALA1908116 | pmol/min/mg protein | Homo sapiens | |||
| 13. | Tamoxifen | Tamoxifen | Km | = | 32 | uM | ALA1908116 | nM | Homo sapiens | |||
| 14. |  Retigabine | 1 (Retigabine) | Km | = | 322 | uM | ALA1908116 | nM | Homo sapiens | |||
| 15. | ALA715 | Olanzapine | Km | = | 227 | uM | ALA1908116 | nM | Homo sapiens | |||
| 16. | ketotifen | ketotifen | Km | = | 86 | uM | ALA1908116 | nM | Homo sapiens | |||
| 17. | ketotifen | ketotifen | Km | = | 59 | uM | ALA1908116 | nM | Homo sapiens | |||
| 18. | Imipramine | Imipramine | Km | = | 310 | uM | ALA1908116 | nM | Homo sapiens | |||
| 19. | α-Hydroxy Tamoxifen | cis-Hydroxy-tamoxifen | Km | = | 101 | uM | ALA1908116 | nM | Homo sapiens | |||
| 20. | α-Hydroxy Tamoxifen | cis-Hydroxy-tamoxifen | Km | = | 95 | uM | ALA1908116 | nM | Homo sapiens |
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