# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | VU 0409106 | 24, VU0409106 | Activity | 0 | ALA2446289 | Not Active | Rattus norvegicus | |||||
2. | ML254 | 38t, VU0430644, ML254 | Activity | 0 | ALA2433903 | Not Active | Rattus norvegicus | |||||
3. | ALA2418364 | 8 | IC50 | = | 3360 | nM | ALA2421150 | 5.47 | nM | Rattus norvegicus | ||
4. | ALA2397347 | 54, VU0469650 | IC50 | > | 10000 | nM | ALA2421150 | nM | Rattus norvegicus | |||
5. | ALA2418364 | 8 | %max | = | 1.1 | % | ALA2421148 | % | Rattus norvegicus | |||
6. | ALA2418365 | 9 | Activity | 0 | ALA2421147 | Not Active | Rattus norvegicus | |||||
7. | ALA2418372 | 16 | Activity | 0 | ALA2421147 | Not Active | Rattus norvegicus | |||||
8. | ALA2338587 | 15c | IC50 | > | 10000 | nM | ALA2343302 | nM | Rattus norvegicus | |||
9. | ALA2338590 | 15f | IC50 | > | 10000 | nM | ALA2343302 | nM | Rattus norvegicus | |||
10. | ALA2338567 | 15w | IC50 | = | 2100 | nM | ALA2343302 | 5.68 | nM | Rattus norvegicus | ||
11. | ALA2338579 | 24d | IC50 | > | 10000 | nM | ALA2343302 | nM | Rattus norvegicus | |||
12. | ALA2338582 | 24g | IC50 | > | 10000 | nM | ALA2343302 | nM | Rattus norvegicus | |||
13. | ALA2338587 | 15c | EC50 | > | 10000 | nM | ALA2343301 | nM | Rattus norvegicus | |||
14. | ALA2338590 | 15f | EC50 | > | 10000 | nM | ALA2343301 | nM | Rattus norvegicus | |||
15. | ALA2338567 | 15w | EC50 | > | 10000 | nM | ALA2343301 | nM | Rattus norvegicus | |||
16. | ALA2338579 | 24d | EC50 | > | 10000 | nM | ALA2343301 | nM | Rattus norvegicus | |||
17. | ALA2338582 | 24g | EC50 | > | 10000 | nM | ALA2343301 | nM | Rattus norvegicus | |||
18. | ALA2011870 | 7, Mixture of trans enantiomers | IC50 | = | 0.9 | nM | ALA2016182 | 9.05 | nM | Rattus norvegicus | ||
19. | ALA3287718 | 67 | Emax | = | 79 | % | ALA3293524 | % | Rattus norvegicus | |||
20. | ALA3287718 | 67 | Emin | = | 3 | % | ALA3293524 | % | Rattus norvegicus |