# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA283758 | X | IC50 | = | 1.9 | uM | ALA675453 | 5.72 | nM | Bos taurus | ||
2. | ALA25553 | II | Inhibition | = | 14 | % | ALA675913 | % | Bos taurus | |||
3. | ALA22509 | V | IC50 | = | 1.5 | uM | ALA675453 | 5.82 | nM | Bos taurus | ||
4. | ALA280917 | III | IC50 | = | 7.4 | uM | ALA675453 | 5.13 | nM | Bos taurus | ||
5. | ALA277199 | VIIIa (diastereoisomer) | IC50 | = | 1.1 | uM | ALA675453 | 5.96 | nM | Bos taurus | ||
6. | ALA281562 | I | IC50 | = | 0.96 | uM | ALA675453 | 6.02 | nM | Bos taurus | ||
7. | ALA25269 | XIIb (diastereoisomer) | Inhibition | = | 31 | % | ALA675454 | % | Bos taurus | |||
8. | Phosphoramidon | Phosphoramidon | IC50 | = | 3.1 | uM | ALA675453 | 5.51 | nM | Bos taurus | ||
9. | ALA277199 | VIIIa (diastereoisomer) | Inhibition | = | 33 | % | ALA675913 | % | Bos taurus | |||
10. | ALA281333 | VI | IC50 | = | 3.4 | uM | ALA675453 | 5.47 | nM | Bos taurus | ||
11. | ALA282663 | XIb (diastereoisomer) | IC50 | = | 3 | uM | ALA675453 | 5.52 | nM | Bos taurus | ||
12. | ALA282663 | XIb (diastereoisomer) | Inhibition | = | 42 | % | ALA675913 | % | Bos taurus | |||
13. | ALA279255 | VII | IC50 | = | 15 | uM | ALA675453 | 4.82 | nM | Bos taurus | ||
14. | ALA277195 | IXa (diastereoisomer) | IC50 | = | 7.1 | uM | ALA675453 | 5.15 | nM | Bos taurus | ||
15. | ALA281785 | IV | IC50 | = | 2.8 | uM | ALA675453 | 5.55 | nM | Bos taurus | ||
16. | ALA25269 | XIIb (diastereoisomer) | IC50 | = | 0.26 | uM | ALA675453 | 6.58 | nM | Bos taurus | ||
17. | ALA277195 | IXa (diastereoisomer) | Inhibition | = | 38 | % | ALA675913 | % | Bos taurus |