# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5276374 | (S)-20a; BGB-8035 | IC50 | = | 61.5 | uM | ALA5251897 | 4.21 | nM | Homo sapiens | ||
2. | ALA5266817 | 50 | INH | 0 | ALA5240419 | Not Active | % | Homo sapiens | ||||
3. | ALA5274179 | 41 | INH | 0 | ALA5240419 | Not Active | % | Homo sapiens | ||||
4. | ALA5266817 | 50 | IC50 | > | 10 | uM | ALA5240413 | nM | Homo sapiens | |||
5. | ALA5274179 | 41 | IC50 | > | 10 | uM | ALA5240413 | nM | Homo sapiens | |||
6. | ALA5274631 | 37 | IC50 | > | 100 | uM | ALA5238212 | nM | Homo sapiens | |||
7. | BI-3406 | I-13 | IC50 | = | 41 | uM | ALA5238212 | 4.39 | nM | Homo sapiens | ||
8. | ALA5282123 | 46 | Activity | > | 100 | % | ALA5237752 | % | Homo sapiens | |||
9. | ALA5278177 | 23 | Activity | > | 100 | % | ALA5237752 | % | Homo sapiens | |||
10. | Soticlestat | SOTICLESTAT | IC50 | = | 14000 | nM | ALA5237308 | 4.85 | nM | Homo sapiens | ||
11. | Imatinib (STI571) | 1 | INH | = | 10 | % | ALA5233747 | % | Homo sapiens | |||
12. | ALA5288115 | 58l | IC50 | = | 50 | uM | ALA5233412 | 4.30 | nM | Homo sapiens | ||
13. | ALA5290158 | 22b | IC50 | = | 7.75 | uM | ALA5233412 | 5.11 | nM | Homo sapiens | ||
14. | ALA5276427 | 22a | IC50 | = | 28.5 | uM | ALA5233412 | 4.54 | nM | Homo sapiens | ||
15. | ALA5275343 | 21a | IC50 | > | 25 | uM | ALA5233412 | nM | Homo sapiens | |||
16. | ALA5270058 | 4; AZD1283 | IC50 | = | 0.399 | uM | ALA5233412 | 6.40 | nM | Homo sapiens | ||
17. | (1R,2S)-2-phenylcyclopropan-1-amine | tranylcypromine | IC50 | = | 14.4 | uM | ALA5232966 | 4.84 | nM | Homo sapiens | ||
18. | ALA5283822 | 10c | IC50 | = | 0.74 | uM | ALA5232966 | 6.13 | nM | Homo sapiens | ||
19. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226241 | nM | Homo sapiens | |||
20. | ALA5276605 | 24 | INH | 0 | ALA5225684 | Not Active | % | Homo sapiens |