# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI-3812 | 44 | % Ctrl | = | 93 | % | ALA5304306 | Not Active | % | Homo sapiens | ||
2. | BI-3802 | BI-3802 | % Ctrl | = | 97 | % | ALA5304203 | Not Active | % | Homo sapiens | ||
3. | ALA3798256 | 6a | Activity | = | 100 | % | ALA3802470 | % | Homo sapiens | |||
4. | LX7101 | 28, LX7101 | INH | > | 90 | % | ALA3801114 | % | Homo sapiens | |||
5. | ALA3792850 | 26 | INH | = | 17.8 | % | ALA3794942 | % | Homo sapiens | |||
6. | ALA3793843 | 24 | INH | = | 43 | % | ALA3794942 | % | Homo sapiens | |||
7. | ALA508964 | 13 | INH | = | 47.3 | % | ALA3794942 | % | Homo sapiens | |||
8. | ALA3775576 | 18 | Activity | = | 11 | % | ALA3777732 | % | Homo sapiens | |||
9. | ALA3774632 | 5b | Activity | >= | 100 | % | ALA3779000 | % | Homo sapiens | |||
10. | ALA3774537 | 54k | INH | 0 | ALA3776419 | Not Active | % | Homo sapiens | ||||
11. | ALA3774885 | 39 | Activity | = | 6 | % | ALA3777732 | % | Homo sapiens | |||
12. | ALA3775317 | 31 | Activity | = | -1 | % | ALA3777732 | % | Homo sapiens | |||
13. | ALA3765499 | 12 | INH | = | 24.9 | % | ALA3767324 | % | Homo sapiens | |||
14. | ALA3758739 | 28 | INH | = | 2.7 | % | ALA3761493 | % | Homo sapiens | |||
15. | ALA3758602 | 15 | INH | = | 10.4 | % | ALA3761294 | % | Homo sapiens | |||
16. | ALA3758502 | 1 | INH | = | 4.3 | % | ALA3761294 | % | Homo sapiens | |||
17. | Cabozantinib (XL184, BMS-907351) | CABOZANTINIB | INH | 0 | ALA3757341 | Not Active | % | Homo sapiens | ||||
18. | ALA3753341 | 6i | INH | 0 | ALA3757340 | Active | % | Homo sapiens | ||||
19. | ALA3753341 | 6i | IC50 | = | 23 | nM | ALA3756062 | 7.64 | nM | Homo sapiens | ||
20. | ALA3753341 | 6i | Activity | = | 5.94 | % | ALA3756051 | % | Homo sapiens |