# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Gemcitabine | Gemzar | CL | = | 0.25 | ml/min/mg | ALA3538245 | mL.min-1.g-1 | Homo sapiens | |||
2. | Gemcitabine | Gemzar | CL | = | 0.35 | ml/min/mg | ALA3538246 | mL.min-1.g-1 | Homo sapiens | |||
3. | Gemcitabine | Gemzar | CL | = | 0.3 | ml/min/mg | ALA3541965 | mL.min-1.g-1 | Homo sapiens | |||
4. | Gemcitabine | Gemzar | Km | = | 610 | uM | ALA3541966 | nM | Homo sapiens | |||
5. | Gemcitabine | Gemzar | Km | = | 562 | uM | ALA3541967 | nM | Homo sapiens | |||
6. | Gemcitabine | Gemzar | Km | = | 630 | uM | ALA3541968 | nM | Homo sapiens | |||
7. | Cytosine β-D-arabinofuranoside | 2 | CL | = | 0.34 | ml/min/mg | ALA3541969 | mL.min-1.g-1 | Homo sapiens | |||
8. | Cytosine β-D-arabinofuranoside | 2 | CL | = | 0.74 | ml/min/mg | ALA3541970 | mL.min-1.g-1 | Homo sapiens | |||
9. | Cytosine β-D-arabinofuranoside | 2 | CL | = | 0.83 | ml/min/mg | ALA3541971 | mL.min-1.g-1 | Homo sapiens | |||
10. | Cytosine β-D-arabinofuranoside | 2 | Km | = | 56 | uM | ALA3541972 | nM | Homo sapiens | |||
11. | Cytosine β-D-arabinofuranoside | 2 | Km | = | 160 | uM | ALA3541973 | nM | Homo sapiens | |||
12. | Cytosine β-D-arabinofuranoside | 2 | Km | = | 138 | uM | ALA3541974 | nM | Homo sapiens | |||
13. | Cytosine β-D-arabinofuranoside | 2 | Vmax | = | 114 | nmol/min/mg | ALA3541974 | nmol/min/mg | Homo sapiens | |||
14. | Cytosine β-D-arabinofuranoside | 2 | Vmax | = | 119 | nmol/min/mg | ALA3541973 | nmol/min/mg | Homo sapiens | |||
15. | Cytosine β-D-arabinofuranoside | 2 | Vmax | = | 19 | nmol/min/mg | ALA3541972 | nmol/min/mg | Homo sapiens | |||
16. | Gemcitabine | Gemzar | Vmax | = | 187 | nmol/min/mg | ALA3541968 | nmol/min/mg | Homo sapiens | |||
17. | Gemcitabine | Gemzar | Vmax | = | 195 | nmol/min/mg | ALA3541967 | nmol/min/mg | Homo sapiens | |||
18. | Gemcitabine | Gemzar | Vmax | = | 151 | nmol/min/mg | ALA3541966 | nmol/min/mg | Homo sapiens | |||
19. | 5,6-Dihydrouridine | 83 (3,4,5,6,-Tetrahydrouridine) | Ki | = | 40 | uM | ALA3241963 | 4.40 | nM | Homo sapiens | ||
20. | ALA1236475 | 5, THU, Epimeric mixture | Ki | = | 440 | uM | ALA3241963 | nM | Homo sapiens |