# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Acelarin (NUC-1031) | 6f, NUC-1031 | Stability | 0 | ALA3132551 | Stable | % | Homo sapiens | ||||
2. | Gemcitabine | Gemzar | Stability | 0 | ALA3132552 | Unstable | % | Homo sapiens | ||||
3. | Tetrahydrouridine | 2b | IC50 | = | 113 | nM | ALA3706053 | 6.95 | 302687 | nM | Homo sapiens | |
4. | ALA3658873 | BDBM159792 | IC50 | = | 140 | nM | ALA3706053 | 6.85 | 302686 | nM | Homo sapiens | |
5. | ALA3658872 | BDBM159791 | IC50 | = | 1616 | nM | ALA3706053 | 5.79 | 302685 | nM | Homo sapiens | |
6. | ALA3658871 | BDBM159790 | IC50 | = | 101 | nM | ALA3706053 | 7.00 | 302684 | nM | Homo sapiens | |
7. | ALA3658870 | BDBM159789 | IC50 | = | 237 | nM | ALA3706053 | 6.62 | 302683 | nM | Homo sapiens | |
8. | ALA3665111 | BDBM111582 | IC50 | = | 2000 | nM | ALA3705845 | 5.70 | 232401 | nM | Homo sapiens | |
9. | ALA3665109 | BDBM111580 | IC50 | = | 4000 | nM | ALA3705845 | 5.40 | 232400 | nM | Homo sapiens | |
10. | ALA3665114 | BDBM111585 | IC50 | = | 400 | nM | ALA3705845 | 6.40 | 232399 | nM | Homo sapiens | |
11. | ALA3665110 | BDBM111581 | IC50 | = | 2000 | nM | ALA3705845 | 5.70 | 232398 | nM | Homo sapiens | |
12. | ALA3665113 | BDBM111584 | IC50 | = | 5000 | nM | ALA3705845 | 5.30 | 232397 | nM | Homo sapiens | |
13. | ALA3665107 | BDBM111578 | IC50 | = | 200 | nM | ALA3705845 | 6.70 | 232396 | nM | Homo sapiens | |
14. | ALA3665108 | BDBM111579 | IC50 | = | 400 | nM | ALA3705845 | 6.40 | 232395 | nM | Homo sapiens | |
15. | ALA3665112 | BDBM111583 | IC50 | = | 5000 | nM | ALA3705845 | 5.30 | 232394 | nM | Homo sapiens | |
16. | ALA3665106 | BDBM111577 | IC50 | = | 400 | nM | ALA3705845 | 6.40 | 232393 | nM | Homo sapiens | |
17. | Gemcitabine | Gemzar | CL | = | 0.25 | ml/min/mg | ALA3538245 | mL.min-1.g-1 | Homo sapiens | |||
18. | Gemcitabine | Gemzar | CL | = | 0.35 | ml/min/mg | ALA3538246 | mL.min-1.g-1 | Homo sapiens | |||
19. | Gemcitabine | Gemzar | CL | = | 0.3 | ml/min/mg | ALA3541965 | mL.min-1.g-1 | Homo sapiens | |||
20. | Gemcitabine | Gemzar | Km | = | 610 | uM | ALA3541966 | nM | Homo sapiens |