# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA363743 | 1 | pKi | = | 7 | ALA5247029 | 7.00 | nM | Homo sapiens | |||
2. | JNJ 10397049 | 9 | pKi | = | 8.3 | ALA5247029 | 8.30 | nM | Homo sapiens | |||
3. | ALA5273790 | 51 | Ki | = | 29 | nM | ALA5244922 | 7.54 | nM | Homo sapiens | ||
4. | ALA3235249 | 1 | Ki | = | 0.2 | nM | ALA5244922 | 9.70 | nM | Homo sapiens | ||
5. | filorexant | FILOREXANT | Ki | = | 0.3 | nM | ALA5244922 | 9.52 | nM | Homo sapiens | ||
6. | ALA3586412 | 4 | Ki | = | 5 | nM | ALA5244922 | 8.30 | nM | Homo sapiens | ||
7. | ALA5174113 | (-)-38; 38b | Ki | = | 34.8 | nM | ALA5243960 | 7.46 | nM | Homo sapiens | ||
8. | ALA5267523 | 26d | Emax | = | 92.3 | % | ALA5243958 | % | Homo sapiens | |||
9. | ALA5281382 | 20c | Emax | = | 2.99 | % | ALA5243958 | % | Homo sapiens | |||
10. | ALA5281062 | 28b | Emax | = | 3.17 | % | ALA5243958 | % | Homo sapiens | |||
11. | ALA5272238 | 31d | Emax | = | 2.89 | % | ALA5243958 | % | Homo sapiens | |||
12. | ALA5278966 | (-)-28d | Emax | = | 97.3 | % | ALA5243958 | % | Homo sapiens | |||
13. | ALA5271252 | (+-)-20d | Emax | = | 171.9 | % | ALA5243958 | % | Homo sapiens | |||
14. | ALA5275698 | 27d | Emax | = | 91.4 | % | ALA5243958 | % | Homo sapiens | |||
15. | ALA5278013 | 20a | Emax | = | 40.2 | % | ALA5243958 | % | Homo sapiens | |||
16. | ALA5282613 | 20b | Emax | = | 2.72 | % | ALA5243958 | % | Homo sapiens | |||
17. | ALA5289437 | 30d | Emax | = | 2.02 | % | ALA5243958 | % | Homo sapiens | |||
18. | ALA5270685 | (-)-20d | Emax | = | 2.59 | % | ALA5243958 | % | Homo sapiens | |||
19. | ALA5278013 | 20a | Emax | = | 105 | % | ALA5243958 | % | Homo sapiens | |||
20. | ALA5287067 | 25d | Emax | = | 61.4 | % | ALA5243958 | % | Homo sapiens |