| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2316207 | 16u | % of control | = | 14 | % | ALA5213515 | % | Homo sapiens | |||
| 2. |  BI 2536 | 1 | % of control | = | 112 | % | ALA5213539 | % | Homo sapiens | |||
| 3. |  ALA4228713 | 22 | % of control | = | 47 | % | ALA5213806 | % | Homo sapiens | |||
| 4. |  ALA4551344 | EUB0000746 | % of control | = | 50 | % | ALA5213987 | % | Homo sapiens | |||
| 5. |  ALA5174953 | 4f | IC50 | = | 805 | nM | ALA5167057 | 6.09 | nM | Homo sapiens | ||
| 6. |  1-[5-tert-butyl-2-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]pyrazol-3-yl]-3-[(1S,4R)-4-[[3-[(2S)-2-methylpiperidin-1-yl]-[1,2,4]triazolo[4,3-a]pyridin-6-yl]oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | 4e | IC50 | = | 944 | nM | ALA5167057 | 6.03 | nM | Homo sapiens | ||
| 7. |  ALA5208103 | 3h | IC50 | = | 2856 | nM | ALA5167057 | 5.54 | nM | Homo sapiens | ||
| 8. |  ALA5197888 | 2m | IC50 | = | 10 | nM | ALA5167057 | 8.00 | nM | Homo sapiens | ||
| 9. |  ALA5184542 | 2h | IC50 | = | 16 | nM | ALA5167057 | 7.80 | nM | Homo sapiens | ||
| 10. |  ALA5206328 | 1c | IC50 | = | 164 | nM | ALA5167057 | 6.79 | nM | Homo sapiens | ||
| 11. |  Nilotinib (AMN-107) | 38 | Activity | 0 | ALA5120259 | Active | Homo sapiens | |||||
| 12. |  ALA3979678 | BDBM238766 | Activity | = | 0.9 | % | ALA4478504 | % | Homo sapiens | |||
| 13. |  ALA4564126 | 18 | INH | <= | 16 | % | ALA4427663 | % | Homo sapiens | |||
| 14. | ALA4564126 | 18 | IC50 | >= | 5 | uM | ALA4427719 | nM | Homo sapiens | |||
| 15. |  JTE-952 | JTE-952; (S)-8b | IC50 | > | 1000 | nM | ALA4424911 | nM | Homo sapiens | |||
| 16. |  8-Anilino-1-naphthalenesulfonic acid | ANS | IC50 | > | 40 | uM | ALA4406950 | nM | Homo sapiens | |||
| 17. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405495 | % | Homo sapiens | |||
| 18. |  ALA4559936 | (+/-)-6 | Activity | = | 5.7 | % | ALA4391485 | % | Homo sapiens | |||
| 19. |  ALA4564973 | 50 | INH | = | 81 | % | ALA4389859 | % | Homo sapiens | |||
| 20. |  ALA4555459 | 43 | INH | = | 68 | % | ALA4389382 | % | Homo sapiens |
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