# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI 653048 | (R)-39 | IC50 | = | 600 | nM | ALA3374308 | 6.22 | nM | Mus musculus | ||
2. | ALA389621 | 12 | t1/2 | = | 60 | min | ALA3281630 | hr | Mus musculus | |||
3. | ALA389621 | 12 | Activity | = | 85 | % | ALA3281635 | % | Mus musculus | |||
4. | ALA3273977 | II, Cort-Alk | INH | 0 | ALA3281641 | Not Active | % | Mus musculus | ||||
5. | ALA389621 | 12 | INH | 0 | ALA3281640 | Not Active | % | Mus musculus | ||||
6. | mechlorethamine | 1 Mechlorethamine | INH | 0 | ALA3281634 | Not Active | % | Mus musculus | ||||
7. | ALA3273977 | II, Cort-Alk | Kd(app) | = | 4.3 | 10'-7M | ALA3281634 | 6.37 | nM | Mus musculus | ||
8. | ALA3273976 | I, Triam Acet-Alk, TA-Alk | Kd(app) | = | 7.5 | 10'-9M | ALA3281634 | 8.12 | nM | Mus musculus | ||
9. | Hydrocortisone phosphate | Hydrocortisone phosphate | INH | 0 | ALA3281632 | Not Active | % | Mus musculus | ||||
10. | ALA389621 | 12 | Kd | = | 4.3 | 10'-8M | ALA3281632 | 7.37 | nM | Mus musculus | ||
11. | Hydrocortisone hydrogen succinate | NSC-7576 | Kd | = | 1.9 | 10'-7M | ALA3281632 | 6.72 | nM | Mus musculus | ||
12. | ALA3273978 | SQ 19435 | INH | 0 | ALA3281632 | Active | % | Mus musculus | ||||
13. | ALA3927299 | 10f | Activity | 0 | ALA3872105 | Active | Mus musculus | |||||
14. | ALA3937005 | 10e | Activity | 0 | ALA3872105 | Active | Mus musculus | |||||
15. | ALA3937406 | 8b | Activity | 0 | ALA3872107 | Mus musculus | ||||||
16. | ALA3956011 | 8c | Activity | 0 | ALA3872107 | Mus musculus | ||||||
17. | ALA3904225 | 8d | Activity | 0 | ALA3872107 | Mus musculus | ||||||
18. | ALA3983602 | 8e | Activity | 0 | ALA3872107 | Mus musculus | ||||||
19. | ALA3954977 | 8f | Activity | 0 | ALA3872107 | Mus musculus | ||||||
20. | ALA3891049 | 8g | Activity | 0 | ALA3872107 | Mus musculus |